SCHEMBL17318481

SCHEMBL17318481

COc1cc(C=CC(=O)c2ccccc2Cl)ccn1

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CXCL12 P48061 5/20 0.61
PTGS1 P23219 2/20 0.55
PTGS2 P35354 2/20 0.55
MAOB P27338 5/20 0.47
MAOA P21397 3/20 0.47
ABCG2 Q9UNQ0 5/20 0.47
ACHE P22303 1/20 0.46
CYP3A4 P08684 1/20 0.46
MAPT P10636 2/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
CASP3 P42574 1/20 0.43
SENP8 Q96LD8 1/20 0.43
SENP7 Q9BQF6 1/20 0.43
SENP6 Q9GZR1 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL363641 0.81 CXCL12 (0.59) CXCL12PTGS1PTGS2MAOBMAOA
SCHEMBL19782926 0.76 CXCL12 (1.00) CXCL12PTGS1PTGS2MAOBMAOA
SCHEMBL25196746 0.76 CXCL12 (0.81) CXCL12PTGS1PTGS2MAOBABCG2
SCHEMBL25245508 0.76 CXCL12 (0.81) CXCL12PTGS1PTGS2MAOBABCG2
SCHEMBL14692575 0.76 MAOB (0.72) CXCL12PTGS1PTGS2MAOBMAOA
SCHEMBL9420986 0.76 MAOB (0.72) CXCL12PTGS1PTGS2MAOBMAOA
SCHEMBL9106499 0.76 TTR (0.54) MAPTALDH1A1LMNACYP2C9CYP2C19
SCHEMBL9106504 0.76 TTR (0.54) MAPTALDH1A1LMNACYP2C9CYP2C19
SCHEMBL30504728 0.75 ABCG2 (0.83) CXCL12PTGS1PTGS2MAOBMAOA
SCHEMBL31448615 0.74 PTGS1 (0.73) CXCL12PTGS1PTGS2MAOBMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015187934-A1 FUNCTIONALIZED HETROARYL ENONES EXHIBITING NRF2 ACTIVATION AND THEIR METHOD OF USE CUREVEDA, LLC (US) 2015-12-10 WO disclosed