SCHEMBL1733696

SCHEMBL1733696

CCN(CC)c1nc(C(N)=O)cc(-c2c(F)cccc2F)n1.Cc1ccccc1-c1cc(C(N)=O)nc(N2CCCCC2)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.48
ALDH1A1 P00352 4/20 0.48
HPGD P15428 4/20 0.48
GAA P10253 2/20 0.48
HSD17B10 Q99714 2/20 0.48
TSHR P16473 1/20 0.48
CASP1 P29466 1/20 0.48
CASP7 P55210 1/20 0.48
TP53 P04637 1/20 0.43
HTT P42858 2/20 0.41
GLA P06280 1/20 0.41
POLB P06746 2/20 0.39
LMNA P02545 1/20 0.39
GPR55 Q9Y2T6 1/20 0.39
MAPK14 Q16539 1/20 0.37
GBA1 P04062 3/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
NPY5R Q15761 2/20 0.34
GRM2 Q14416 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1734174 0.82 ALDH1A1 (0.70) KDM4EALDH1A1HPGDGAAHSD17B10
SCHEMBL1733748 0.80 KDM4E (0.70) KDM4EALDH1A1HPGDHTTGPR55
SCHEMBL1734432 0.80 KDM4E (0.67) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL1733464 0.78 KDM4E (0.70) KDM4EALDH1A1HPGDGAAHSD17B10
SCHEMBL1733617 0.77 KDM4E (0.69) KDM4ELMNAGRM2ADORA2AADORA1
SCHEMBL3724502 0.77 KDM4E (0.54) KDM4EALDH1A1HPGDGAAHSD17B10
SCHEMBL1733755 0.76 KDM4E (0.63) KDM4EALDH1A1HPGDGAAHSD17B10
SCHEMBL1734590 0.76 KDM4E (0.63) KDM4EALDH1A1HPGDGAAHSD17B10
SCHEMBL1733665 0.74 KDM4E (0.64) KDM4EMEN1KMT2AGRM2ADORA2A
SCHEMBL3720267 0.74 KDM4E (0.55) KDM4EALDH1A1HPGDGAAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1891018-B1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMA (US) 2011-11-16 EP claimed
WO-2011131686-A1 A THERMALLY CONTROLLED ASSEMBLY NAPATECH A/S (DK) 2011-10-27 WO claimed