SCHEMBL17338995

SCHEMBL17338995

O=C1C2C(c3ccc(Br)cc3)[C@@H]2C(=O)N1c1cc(Cl)cc(Cl)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGAL P20701 9/20 0.42
ITGB2 P05107 8/20 0.41
ICAM1 P05362 8/20 0.41
ATM Q13315 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CNR1 P21554 1/20 0.38
ALOX15 P16050 2/20 0.37
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
ALOX12 P18054 1/20 0.37
KMT2A Q03164 1/20 0.37
HSD17B10 Q99714 1/20 0.37
ADCY2 Q08462 1/20 0.36
CYP3A4 P08684 3/20 0.36
CYP2C9 P11712 3/20 0.36
CYP2C19 P33261 2/20 0.36
LMNA P02545 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17338998 1.00 ITGAL (0.42) ITGALITGB2ICAM1ATML3MBTL1
SCHEMBL18787390 1.00 ITGAL (0.42) ITGALITGB2ICAM1ATML3MBTL1
SCHEMBL17338997 1.00 ITGAL (0.42) ITGALITGB2ICAM1ATML3MBTL1
SCHEMBL17347096 1.00 ITGAL (0.42) ITGALITGB2ICAM1ATML3MBTL1
SCHEMBL17347061 1.00 ITGAL (0.42) ITGALITGB2ICAM1ATML3MBTL1
SCHEMBL17347068 0.83 ALDH1A1 (0.48) ATMALOX15MEN1ALDH1A1GAA
SCHEMBL22898500 0.83 ALDH1A1 (0.48) ATMALOX15MEN1ALDH1A1GAA
SCHEMBL17347124 0.83 ALDH1A1 (0.48) ATMALOX15MEN1ALDH1A1GAA
SCHEMBL17338881 0.83 ALDH1A1 (0.48) ATMALOX15MEN1ALDH1A1GAA
SCHEMBL18787456 0.83 ALDH1A1 (0.48) ATMALOX15MEN1ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3154941-A1 SMALL MOLECULE LFA-1 INHIBITORS AlloCyte Pharmaceuticals AG (CH) 2017-04-19 EP disclosed
WO-2015189265-A1 SMALL MOLECULE LFA-1 INHIBITORS ALLOCYTE PHARMACEUTICALS AG (CH) 2015-12-17 WO disclosed