SCHEMBL17340288

SCHEMBL17340288

CSc1nc(Cl)c(C(N)=O)c(Nc2cccc(S(=O)(=O)N(N)N)c2)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 6/20 0.47
CA2 P00918 6/20 0.47
CA7 P43166 5/20 0.47
CA13 Q8N1Q1 4/20 0.43
PPARG P37231 2/20 0.37
CDK1 P06493 2/20 0.37
CDK2 P24941 2/20 0.37
CCNB2 O95067 1/20 0.37
CCNE2 O96020 1/20 0.37
CCNB1 P14635 1/20 0.37
CCNE1 P24864 1/20 0.37
CCNB3 Q8WWL7 1/20 0.37
ALK Q9UM73 3/20 0.37
EGFR P00533 2/20 0.37
BTK Q06187 2/20 0.37
CDC7 O00311 1/20 0.37
PLK4 O00444 1/20 0.37
CHEK1 O14757 1/20 0.37
AURKA O14965 1/20 0.37
DCLK1 O15075 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10156677 0.92 CCNB2 (0.45) CA1CA2CA7CA13CDK1
SCHEMBL10127055 0.89 CA1 (0.52) CA1CA2CA7CA13CDK1
SCHEMBL282561 0.89 ALK (0.46) CA1CA2CA7CA13PPARG
SCHEMBL10127071 0.87 CA1 (0.43) CA1CA2CA7CA13PPARG
SCHEMBL10156697 0.87 TNNI3K (0.48) CA1CA2CA7EGFRTNNI3K
SCHEMBL10127073 0.86 CA1 (0.42) CA1CA2CA7CA13PPARG
SCHEMBL10156701 0.85 CA1 (0.41) CA1CA2CA7CA13PPARG
SCHEMBL10127040 0.82 TP53 (0.46) PPARGCDK1CDK2CCNB2CCNE2
SCHEMBL17069444 0.82 LMNA (0.47) PPARGEGFRFERKDRSYK
SCHEMBL10127045 0.80 MAPT (0.45) CA1CA2CA7PPARGKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2428508-B1 DIAMINO HETEROCYCLIC CARBOXAMIDE COMPOUND ASTELLAS PHARMA INC (JP) 2015-12-16 EP disclosed