SCHEMBL17340682

SCHEMBL17340682

C=C(NC)c1c(-c2ccc(F)cc2)oc2ccc(-c3cccc(C(=O)N[C@@H](CO)c4ccccc4)c3)cc12

nearest known ligand 0.47

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 10/20 0.47
ROCK1 Q13464 6/20 0.47
CYP3A4 P08684 1/20 0.43
CYP2C8 P10632 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10241939 0.93 CYP3A4 (0.51) ROCK2ROCK1CYP3A4CYP2C8
SCHEMBL10241977 0.86 CYP3A4 (0.49) ROCK2ROCK1CYP3A4CYP2C8
SCHEMBL17340649 0.82 CYP3A4 (0.42) CYP3A4CYP2C8
SCHEMBL17340648 0.82 HPGDS (0.45) ROCK2CYP3A4CYP2C8
SCHEMBL10240167 0.81 CYP3A4 (0.53) ROCK2CYP3A4CYP2C8
SCHEMBL10280748 0.81 CYP3A4 (0.50) ROCK2ROCK1CYP3A4CYP2C8
SCHEMBL10280771 0.79 CYP3A4 (0.48) CYP3A4CYP2C8
SCHEMBL10242010 0.79 CYP3A4 (0.48) ROCK2ROCK1CYP3A4CYP2C8
SCHEMBL10241946 0.78 CYP3A4 (0.49) ROCK2ROCK1CYP3A4CYP2C8
SCHEMBL10242000 0.78 CYP3A4 (0.49) ROCK2ROCK1CYP3A4CYP2C8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2326633-B1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL MYERS SQUIBB CO (US) 2015-12-16 EP disclosed