SCHEMBL1734368

SCHEMBL1734368

CCN(CC)c1nc(C(N)=O)cc(-c2cccc(NC(C)=O)c2)n1.CN(CCc1c[nH]c2ccccc12)c1nc(C(N)=O)cc(-c2ccccc2)n1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.53
AKT1 P31749 1/20 0.42
CDK4 P11802 8/20 0.42
CCND1 P24385 8/20 0.42
CDK2 P24941 2/20 0.42
MAPT P10636 2/20 0.40
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
ALDH1A1 P00352 2/20 0.39
PARP1 P09874 1/20 0.39
DHODH Q02127 1/20 0.39
MOK Q9UQ07 2/20 0.39
ABCB1 P08183 1/20 0.39
ABCC1 P33527 1/20 0.39
ABCG2 Q9UNQ0 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
HTR1A P08908 1/20 0.38
ADRA2A P08913 1/20 0.38
ADRA2B P18089 1/20 0.38
ADRA2C P18825 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1733586 0.87 KDM4E (0.53) KDM4ECDK4CCND1CDK2HTR1A
SCHEMBL1734451 0.81 KDM4E (0.69) KDM4EMAPTMEN1KMT2AALDH1A1
SCHEMBL1733607 0.73 KDM4E (1.00) KDM4EMAPTMEN1KMT2AALDH1A1
SCHEMBL1733450 0.70 KDM4E (0.64) KDM4EALDH1A1
SCHEMBL1734567 0.70 KDM4E (0.78) KDM4EMEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL1733742 0.69 KDM4E (0.85) KDM4EMEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL1733611 0.68 KDM4E (0.83) KDM4EMEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL1733590 0.68 HTR1A (0.48) CDK4CCND1MEN1KMT2AALDH1A1
SCHEMBL1734118 0.67 KDM4E (0.66) KDM4EMEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL1733610 0.67 KDM4E (0.81) KDM4EMEN1KMT2AALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1891018-B1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMA (US) 2011-11-16 EP claimed
WO-2011131686-A1 A THERMALLY CONTROLLED ASSEMBLY NAPATECH A/S (DK) 2011-10-27 WO claimed