SCHEMBL17347163

SCHEMBL17347163

Cc1cc(C)cc(N2C(=O)[C@@H]3[C@H](c4ccc(Br)cc4)[C@]3(C)C2=O)c1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADCY2 Q08462 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
CACNA1B Q00975 2/20 0.38
APBA1 Q02410 2/20 0.38
NPSR1 Q6W5P4 1/20 0.37
ITGAL P20701 4/20 0.36
ITGB2 P05107 3/20 0.36
ICAM1 P05362 3/20 0.36
HSP90AA1 P07900 1/20 0.36
CCR6 P51684 1/20 0.36
HSD11B1 P28845 2/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17347161 1.00 ADCY2 (0.41) ADCY2MEN1KMT2ACACNA1BAPBA1
SCHEMBL17347069 0.88 ITGAL (0.48) ITGALITGB2ICAM1
SCHEMBL22898547 0.88 ITGAL (0.48) ITGALITGB2ICAM1
SCHEMBL22898584 0.88 ITGAL (0.48) ITGALITGB2ICAM1
SCHEMBL17347097 0.88 ITGAL (0.48) ITGALITGB2ICAM1
SCHEMBL17347215 0.88 ITGAL (0.48) ITGALITGB2ICAM1
SCHEMBL18787389 0.88 ITGAL (0.48) ITGALITGB2ICAM1
SCHEMBL17347160 0.86 ADCY2 (0.45) ADCY2MEN1KMT2ACACNA1BAPBA1
SCHEMBL17347156 0.86 ADCY2 (0.45) ADCY2MEN1KMT2ACACNA1BAPBA1
SCHEMBL17347392 0.83 ITGAL (0.39) ADCY2CACNA1BAPBA1NPSR1ITGAL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015189265-A1 SMALL MOLECULE LFA-1 INHIBITORS ALLOCYTE PHARMACEUTICALS AG (CH) 2015-12-17 WO disclosed