SCHEMBL1734847

SCHEMBL1734847

CC(C)(C)N(C(=O)O)c1ccc(-c2nc3cc(C#N)cc(CBr)c3o2)cc1

nearest known ligand 0.46

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.46
ESR2 Q92731 1/20 0.46
CEPT1 Q9Y6K0 10/20 0.44
CETP P11597 10/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1733937 0.86 CEPT1 (0.53) CEPT1CETP
SCHEMBL1734955 0.85 CEPT1 (0.44) CEPT1CETP
SCHEMBL4526793 0.81 CEPT1 (0.54) ESR1ESR2CEPT1CETP
SCHEMBL17512330 0.68 KMT2A (0.41)
SCHEMBL1735035 0.68 CEPT1 (0.70) CEPT1CETP
SCHEMBL3681612 0.68 ESR2 (0.55) ESR1ESR2CEPT1CETP
SCHEMBL4531439 0.68 CEPT1 (0.68) CEPT1CETP
SCHEMBL3746100 0.67 ESR2 (0.52) ESR1ESR2CEPT1CETP
SCHEMBL2837210 0.67 CETP (0.50) ESR1ESR2CEPT1CETP
SCHEMBL3807420 0.67 CETP (0.64) CEPT1CETP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1954287-B1 CETP INHIBITORS MERCK SHARP & DOHME (US) 2011-11-16 EP disclosed
US-20110262658-A1 PROCESS AND DEVICE FOR TREATING THE COATING OF THERMOPLASTIC RESIN CONTAINERS ZOPPAS MATTEO 2011-10-27 US disclosed