SCHEMBL1735289

SCHEMBL1735289

CCN(CC)CCOc1ccc(Nc2ncc(-c3ccc(CC(=O)O)cc3)cn2)cc1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 5/20 0.50
CDK4 P11802 5/20 0.50
CCND1 P24385 5/20 0.50
CCND2 P30279 5/20 0.50
CCND3 P30281 5/20 0.50
RIPK2 O43353 7/20 0.49
NOD2 Q9HC29 7/20 0.49
ACVR1 Q04771 5/20 0.49
WEE1 P30291 1/20 0.45
CYP1A2 P05177 1/20 0.44
LTA4H P09960 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
HTT P42858 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1734414 0.88 CDK4 (0.47) MCHR1CDK4CCND1CCND2CCND3
SCHEMBL1735255 0.87 CSNK2A1 (0.60) MCHR1CDK4CCND1CCND2CCND3
SCHEMBL1735178 0.85 MCHR1 (0.52) MCHR1CDK4CCND1CCND2CCND3
SCHEMBL13605301 0.85 RIPK2 (0.61) MCHR1CDK4CCND1CCND2CCND3
SCHEMBL13605344 0.84 CDK4 (0.54) MCHR1CDK4CCND1CCND2CCND3
SCHEMBL1735257 0.84 MCHR1 (0.59) MCHR1CDK4CCND1CCND2CCND3
SCHEMBL1734406 0.83 MCHR1 (0.65) MCHR1CDK4CCND1CCND2CCND3
SCHEMBL1734426 0.83 MCHR1 (0.54) MCHR1CDK4CCND1CCND2CCND3
SCHEMBL1734211 0.82 RARA (0.52) MCHR1CDK4CCND1CCND2CCND3
SCHEMBL4212893 0.82 CYP1A2 (0.63) CYP1A2LTA4HCYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1928236-B1 DIARYLAMINE-CONTAINING COMPOUNDS AND COMPOSITIONS, AND THEIR USE AS MODULATORS OF C-KIT RECEPTORS IRM LLC (BM) 2011-11-23 EP claimed