SCHEMBL17354366

SCHEMBL17354366

Cc1ccccc1NC(=O)Nc1nc(=O)c(-c2ccc(CNCCCN)cc2C)c[nH]1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MC4R P32245 3/20 0.38
MC5R P33032 2/20 0.38
MC3R P41968 2/20 0.38
DDX3X O00571 2/20 0.36
IMPDH2 P12268 2/20 0.36
KMT2A Q03164 2/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
ITGB1 P05556 4/20 0.36
ITGA4 P13612 4/20 0.36
KDR P35968 2/20 0.34
MC1R Q01726 2/20 0.34
GAA P10253 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
PDGFRB P09619 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17354368 0.93 MC4R (0.37) MC4RMC5RMC3RDDX3XIMPDH2
SCHEMBL17354133 0.91 KDR (0.41) DDX3XIMPDH2KMT2AKDM4EMEN1
SCHEMBL17486587 0.89 IGF1R (0.36) MC4RMC5RMC3RKMT2AMEN1
SCHEMBL13677 0.88 IDH1 (0.37) MC4RMC5RMC3RITGB1ITGA4
SCHEMBL17354281 0.85 PDCD1LG2 (0.36) MC4RMC5RMC3RKDR
SCHEMBL17354195 0.84 PTGER3 (0.37) DDX3XIMPDH2ITGB1ITGA4KDR
SCHEMBL17354162 0.84 KDR (0.36) DDX3XIMPDH2KMT2AKDM4EMEN1
SCHEMBL17354138 0.84 KDR (0.42) DDX3XIMPDH2KMT2AKDM4EMEN1
SCHEMBL17354348 0.84 KDR (0.37) DDX3XIMPDH2KMT2AKDM4EMEN1
SCHEMBL17354370 0.83 HDAC3 (0.36) MC4RMC5RMC3R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9216979-B2 Antimicrobial compounds and methods of making and using the same MELINTA THERAPEUTICS, INC. (US) 2015-12-22 US disclosed