SCHEMBL17354476

SCHEMBL17354476

CSCCNCc1ccc(-c2c[nH]c(NC(=O)Nc3ccccc3OCF)nc2=O)cc1Cl

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.36
NPC1 O15118 2/20 0.34
RAB9A P51151 1/20 0.34
KMT2A Q03164 3/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
MEN1 O00255 2/20 0.34
ALDH1A1 P00352 1/20 0.34
CHEK1 O14757 2/20 0.34
MAPT P10636 4/20 0.33
IGF1R P08069 6/20 0.33
PDCD1LG2 Q9BQ51 1/20 0.32
CD274 Q9NZQ7 1/20 0.32
HTR3E A5X5Y0 1/20 0.32
HTR3B O95264 1/20 0.32
HTR3A P46098 1/20 0.32
HTR3D Q70Z44 1/20 0.32
HTR3C Q8WXA8 1/20 0.32
ROCK2 O75116 1/20 0.32
LIMK1 P53667 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17354489 0.90 ABL1 (0.38)
SCHEMBL17486551 0.90 IGF1R (0.35) LMNANPC1RAB9AKMT2ASMN1; SMN2
SCHEMBL17354480 0.89 IGF1R (0.36) LMNANPC1RAB9AKMT2ASMN1; SMN2
SCHEMBL14853463 0.84 HTT (0.32) KMT2AMEN1ALDH1A1CHEK1MAPT
SCHEMBL17354473 0.82 IGF1R (0.37) CHEK1IGF1RROCK2LIMK1
SCHEMBL13725 0.81 IDH2 (0.38) IGF1R
SCHEMBL14853169 0.81 RAB9A (0.38) NPC1RAB9AKMT2ASMN1; SMN2MEN1
SCHEMBL17354144 0.80 PTGER3 (0.37) ALDH1A1MAPT
SCHEMBL14075 0.79 KIT (0.38)
SCHEMBL13706 0.79 KIT (0.38) IGF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9216979-B2 Antimicrobial compounds and methods of making and using the same MELINTA THERAPEUTICS, INC. (US) 2015-12-22 US disclosed