SCHEMBL17355225

SCHEMBL17355225

COc1cccc(-c2ccc3c(c2)C(=O)C2(CCCCC2)C3)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 3/20 0.47
CHEK1 O14757 1/20 0.43
BACE1 P56817 3/20 0.43
ALKBH3 Q96Q83 1/20 0.43
NCOA1 Q15788 1/20 0.42
NCOA3 Q9Y6Q9 1/20 0.42
BRD4 O60885 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
FGFR1 P11362 1/20 0.40
HTR1A P08908 2/20 0.39
ADRA2A P08913 1/20 0.39
ADRA2B P18089 1/20 0.39
ADRA2C P18825 1/20 0.39
DRD4 P21917 1/20 0.39
SLC6A2 P23975 1/20 0.39
HTR2C P28335 1/20 0.39
SLC6A4 P31645 1/20 0.39
OPRK1 P41145 1/20 0.39
HTR2B P41595 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7889463 0.89 PGR (0.46) PGRCHEK1BACE1ALKBH3NCOA1
SCHEMBL12748158 0.87 PGR (0.47) PGRCHEK1BACE1ALKBH3NCOA1
SCHEMBL12747661 0.87 BACE1 (0.45) PGRCHEK1BACE1ALKBH3NCOA1
SCHEMBL12748135 0.83 BACE1 (0.56) PGRCHEK1BACE1ALKBH3NCOA1
SCHEMBL7892335 0.83 BACE1 (0.56) PGRCHEK1BACE1ALKBH3NCOA1
SCHEMBL12748238 0.81 BACE1 (0.53) PGRCHEK1BACE1ALKBH3NCOA1
SCHEMBL12748242 0.80 BACE1 (0.55) PGRCHEK1BACE1ALKBH3NCOA1
SCHEMBL30483 0.78 BACE1 (0.59) PGRCHEK1BACE1
SCHEMBL12746120 0.78 BACE1 (0.44) PGRBACE1SLC6A2SLC6A4SLC6A3
SCHEMBL7888134 0.77 PGR (0.44) PGRCHEK1ALKBH3NCOA1NCOA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2406240-B1 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS INC (US) 2015-12-23 EP disclosed