SCHEMBL17360615

SCHEMBL17360615

O=C(c1ccccc1)c1ccccc1CN1C(=O)c2ccccc2C1(O)c1ccc(Cl)cc1

nearest known ligand 0.68

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MDM2 Q00987 17/20 0.68
CYP2D6 P10635 2/20 0.57
CYP3A4 P08684 1/20 0.57
TP53 P04637 1/20 0.49
RAF1 P04049 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12305425 0.86 MDM2 (0.82) MDM2CYP2D6CYP3A4
SCHEMBL1828449 0.86 MDM2 (0.82) MDM2CYP2D6CYP3A4
SCHEMBL1819888 0.81 MDM2 (1.00) MDM2CYP2D6CYP3A4RAF1
SCHEMBL15863686 0.81 MDM2 (0.73) MDM2CYP2D6CYP3A4TP53RAF1
SCHEMBL1819470 0.80 MDM2 (1.00) MDM2CYP2D6CYP3A4
SCHEMBL7995300 0.79 MDM2 (1.00) MDM2CYP2D6CYP3A4RAF1
SCHEMBL2457547 0.79 MDM2 (1.00) MDM2CYP2D6CYP3A4RAF1
SCHEMBL7989560 0.77 MDM2 (1.00) MDM2CYP2D6CYP3A4TP53
SCHEMBL2459937 0.77 MDM2 (1.00) MDM2CYP2D6CYP3A4TP53
SCHEMBL2455286 0.75 MDM2 (0.88) MDM2CYP2D6CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2960233-A1 NEW THERAPEUTIC AGENTS Cancer Research Technology Limited (GB) 2015-12-30 EP disclosed