SCHEMBL17364461

SCHEMBL17364461

Cc1c(C(=O)C(C)C)c(N)nn1-c1cccc(Cl)c1F

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.45
RIPK1 Q13546 2/20 0.41
PDE4B Q07343 1/20 0.40
MDM2 Q00987 10/20 0.37
MDM4 O15151 8/20 0.37
WNT3A P56704 1/20 0.35
LMNA P02545 1/20 0.35
P2RX7 Q99572 1/20 0.35
HDAC9 Q9UKV0 1/20 0.35
NPSR1 Q6W5P4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17365310 0.86 RIPK1 (0.46) NOTUMRIPK1PDE4BMDM2MDM4
SCHEMBL17563304 0.86 NOTUM (0.51) NOTUMRIPK1PDE4BMDM2WNT3A
SCHEMBL15930179 0.86 RIPK1 (0.48) NOTUMRIPK1PDE4BMDM2MDM4
SCHEMBL18945160 0.76 NOTUM (0.48) NOTUMRIPK1PDE4BMDM2MDM4
SCHEMBL15930148 0.76 SCN9A (0.43) NOTUMRIPK1MDM2LMNAHDAC9
SCHEMBL15930147 0.76 NOTUM (0.47) NOTUMRIPK1HDAC9NPSR1
SCHEMBL15930146 0.76 NOTUM (0.44) NOTUMRIPK1MDM2LMNA
SCHEMBL15933281 0.75 NPSR1 (0.52) NOTUMRIPK1PDE4BMDM2WNT3A
SCHEMBL20209694 0.75 RIPK1 (0.45) NOTUMRIPK1PDE4BMDM2MDM4
SCHEMBL15930151 0.75 NOTUM (0.41) NOTUMRIPK1MDM2MDM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9221818-B2 Macrocycles as factor XIa inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2015-12-29 US disclosed