SCHEMBL173715

SCHEMBL173715

O=S(=O)(c1ccc(Cn2ccnc2)cc1)c1cccc(-n2cccn2)c1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 3/20 0.54
CYP11B1 P15538 6/20 0.45
CYP11B2 P19099 6/20 0.45
CYP19A1 P11511 4/20 0.45
CYP1A2 P05177 1/20 0.44
POLB P06746 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
MAPT P10636 1/20 0.44
TBXAS1 P24557 1/20 0.44
QPCT Q16769 1/20 0.44
CYP4Z1 Q86W10 1/20 0.44
QPCTL Q9NXS2 1/20 0.44
CYP17A1 P05093 1/20 0.43
CYP2A6 P11509 1/20 0.43
CYP2B6 P20813 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL164101 0.83 CYP11B1 (0.47) CYP11B1CYP11B2CYP19A1CYP1A2POLB
SCHEMBL21500650 0.83 NAMPT (0.56) NAMPTCYP11B1CYP11B2CYP19A1CYP1A2
SCHEMBL21500639 0.83 NAMPT (0.56) NAMPTCYP11B1CYP11B2CYP19A1CYP1A2
SCHEMBL159804 0.82 CYP11B1 (0.47) CYP11B1CYP11B2CYP17A1
SCHEMBL21500648 0.81 NAMPT (0.55) NAMPTCYP11B1CYP11B2CYP19A1CYP1A2
SCHEMBL22399251 0.81 NAMPT (0.58) NAMPTCYP19A1POLB
SCHEMBL19742865 0.80 CYP11B1 (0.68) CYP11B1CYP11B2CYP19A1CYP1A2POLB
SCHEMBL22399257 0.80 NAMPT (0.51) NAMPTCYP11B1CYP19A1CYP3A4CYP17A1
SCHEMBL22399266 0.77 CYP11B1 (0.51) CYP11B1CYP11B2CYP19A1CYP1A2POLB
SCHEMBL21500662 0.77 NAMPT (0.49) NAMPTCYP11B1CYP11B2CYP19A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2611804-A1 NOVEL COMPOUNDS AND COMPOSITIONS FOR THE INHIBITION OF NAMPT Forma TM, LLC. (US) 2013-07-10 EP disclosed
WO-2012031197-A1 NOVEL COMPOUNDS AND COMPOSITIONS FOR THE INHIBITION OF NAMPT FORMA THERAPEUTICS, INC. (US) 2012-03-08 WO disclosed