SCHEMBL17375008

SCHEMBL17375008

COc1c(C(C)(C)C)cc(N2CCC(=O)NC2=O)c(F)c1/C=C/c1ccc(NS(C)(=O)=O)cc1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.47
CRBN Q96SW2 2/20 0.37
TRPV1 Q8NER1 1/20 0.33
DDB1 Q16531 1/20 0.32
TDP2 O95551 1/20 0.31
PIP4K2A P48426 2/20 0.30
PIP4K2B P78356 2/20 0.30
NR3C2 P08235 1/20 0.30
AURKB Q96GD4 1/20 0.30
TNFRSF1A P19438 1/20 0.30
HTR7 P34969 1/20 0.30
HTR6 P50406 1/20 0.30
ABCB1 P08183 1/20 0.30
KIF11 P52732 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17375076 0.88 CYP3A4 (0.36) CYP3A4CRBNDDB1
SCHEMBL17378859 0.86 CRBN (0.38) CYP3A4CRBNDDB1AURKBHTR7
SCHEMBL17378945 0.86 CYP3A4 (0.36) CYP3A4CRBNDDB1AURKB
SCHEMBL1530350 0.83 CYP3A4 (0.56) CYP3A4CRBNTRPV1DDB1TDP2
SCHEMBL1530351 0.83 CYP3A4 (0.56) CYP3A4CRBNTRPV1DDB1TDP2
SCHEMBL1530391 0.83 CYP3A4 (0.56) CYP3A4CRBNTRPV1DDB1TDP2
SCHEMBL17378791 0.83 CRBN (0.36) CYP3A4CRBNDDB1TDP2
SCHEMBL17375035 0.81 CRBN (0.50) CYP3A4CRBNDDB1TDP2NR3C2
SCHEMBL17378862 0.79 CRBN (0.38) CRBNDDB1
SCHEMBL17375001 0.78 GAA (0.36) CYP3A4CRBNDDB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015197028-A1 COMPOUNDS AS HEPATITIS C VIRUS (HCV) INHIBITORS AND USES THEREOF IN MEDICINE SUNSHINE LAKE PHARMA CO., LTD. (CN) 2015-12-30 WO disclosed
WO-2015197028-A1 COMPOUNDS AS HEPATITIS C VIRUS (HCV) INHIBITORS AND USES THEREOF IN MEDICINE SUNSHINE LAKE PHARMA CO., LTD. (CN) 2015-12-30 WO disclosed