SCHEMBL1738176

SCHEMBL1738176

CCOC(=O)C1CCN(CCc2ccc(-c3noc(-c4nn(CC)cc4-c4ccccc4)n3)cc2C(F)(F)F)CC1

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
KDM4E B2RXH2 2/20 0.43
S1PR1 P21453 14/20 0.42
S1PR3 Q99500 5/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1740595 0.92 S1PR1 (0.49) S1PR1S1PR3
SCHEMBL1739327 0.85 ALDH1A1 (0.43) ALDH1A1SMN1; SMN2KDM4ES1PR1S1PR3
SCHEMBL1738177 0.79 S1PR1 (0.41) ALDH1A1SMN1; SMN2KDM4ES1PR1S1PR3
SCHEMBL1739399 0.78 ALDH1A1 (0.47) ALDH1A1SMN1; SMN2KDM4ES1PR1S1PR3
SCHEMBL1739595 0.78 ALDH1A1 (0.45) ALDH1A1SMN1; SMN2KDM4ES1PR1S1PR3
SCHEMBL1740182 0.78 ALDH1A1 (0.45) ALDH1A1SMN1; SMN2KDM4ES1PR1S1PR3
SCHEMBL1741103 0.78 S1PR1 (0.46) S1PR1S1PR3
SCHEMBL12154424 0.77 S1PR1 (0.38) ALDH1A1SMN1; SMN2KDM4ES1PR1S1PR3
SCHEMBL1739720 0.75 S1PR1 (0.48) S1PR1S1PR3
SCHEMBL1740694 0.72 S1PR1 (0.48) S1PR1S1PR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2390252-A1 New pyrazole derivatives Almirall, S.A. (ES) 2011-11-30 EP disclosed
EP-2390252-A1 New pyrazole derivatives Almirall, S.A. (ES) 2011-11-30 EP disclosed
WO-2011144338-A1 PYRAZOLE DERIVATIVES AS S1P1 AGONISTS ALMIRALL, S.A. (ES) 2011-11-24 WO disclosed
WO-2011144338-A1 PYRAZOLE DERIVATIVES AS S1P1 AGONISTS ALMIRALL, S.A. (ES) 2011-11-24 WO disclosed