SCHEMBL17383003

SCHEMBL17383003

COc1cc(C)[nH]c(=O)c1CN1CCc2c(C)cc(-c3c(C)noc3C)c(Cl)c2C1=O

nearest known ligand 0.89

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
EZH2 Q15910 20/20 0.89
EZH1 Q92800 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17382971 0.94 EZH2 (1.00) EZH2EZH1
SCHEMBL29408704 0.86 EZH2 (1.00) EZH2
SCHEMBL29408702 0.86 EZH2 (1.00) EZH2
SCHEMBL15813960 0.86 EZH2 (1.00) EZH2
SCHEMBL22645619 0.84 EZH2 (0.75) EZH2
SCHEMBL29840768 0.84 EZH2 (0.75) EZH2
SCHEMBL17382510 0.83 EZH2 (0.79) EZH2EZH1
SCHEMBL22645641 0.83 EZH2 (1.00) EZH2
SCHEMBL22645622 0.83 EZH2 (0.75) EZH2EZH1
SCHEMBL29840778 0.83 EZH2 (0.75) EZH2EZH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015193768-A1 ARYL FUSED LACTAMS AS EZH2 MODULATORS PFIZER INC. (US) 2015-12-23 WO disclosed