SCHEMBL1738508

SCHEMBL1738508

CCOC(=O)C(=O)CC(=O)c1ccccc1OC

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.59
IDO1 P14902 1/20 0.56
TDO2 P48775 1/20 0.56
KMT2A Q03164 2/20 0.55
LMNA P02545 2/20 0.55
MAPT P10636 2/20 0.55
MEN1 O00255 1/20 0.55
PLIN1 O60240 1/20 0.55
POLB P06746 1/20 0.55
PLIN5 Q00G26 1/20 0.55
ABHD5 Q8WTS1 1/20 0.55
GAA P10253 1/20 0.52
CTSD P07339 1/20 0.51
ALDH1A1 P00352 1/20 0.50
HTT P42858 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
CYP19A1 P11511 1/20 0.50
HDAC8 Q9BY41 1/20 0.49
HDAC1 Q13547 1/20 0.49
RAB9A P51151 4/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31039791 1.00 NPC1 (0.59) NPC1IDO1TDO2KMT2ALMNA
SCHEMBL29819654 0.87 NPC1 (0.66) NPC1IDO1TDO2KMT2ALMNA
SCHEMBL20239567 0.87 NPC1 (0.66) NPC1IDO1TDO2KMT2ALMNA
SCHEMBL17114470 0.86 NPC1 (0.64) NPC1IDO1TDO2KMT2ALMNA
SCHEMBL17114471 0.86 NPC1 (0.64) NPC1IDO1TDO2KMT2ALMNA
SCHEMBL954173 0.84 NPC1 (0.62) NPC1IDO1TDO2KMT2ALMNA
SCHEMBL30218361 0.84 NPC1 (0.62) NPC1IDO1TDO2KMT2ALMNA
SCHEMBL18304687 0.84 HPGD (0.49) NPC1KMT2ALMNAMAPTMEN1
SCHEMBL17317414 0.83 TSHR (0.52) NPC1KMT2ALMNAMAPTMEN1
SCHEMBL1739513 0.83 ERCC5 (0.65) NPC1KMT2ALMNAMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12325702-B2 ATF6 inhibitors and uses thereof ALTOS LABS, INC. (US) 2025-06-10 US disclosed
US-20240124434-A1 ATF6 INHIBITORS AND USES THEREOF ALTOS LABS, INC. 2024-04-18 US disclosed
US-20210221803-A1 ATF6 INHIBITORS AND USES THEREOF ALTOS LABS, INC. 2021-07-22 US disclosed
US-20210221803-A1 ATF6 INHIBITORS AND USES THEREOF ALTOS LABS, INC. 2021-07-22 US disclosed
EP-3774782-A2 ATF6 INHIBITORS AND USES THEREOF Black Belt TX Ltd (GB) 2021-02-17 EP disclosed
CN-112313224-A ATF6 inhibitors and uses thereof 黑带医疗有限责任公司 2021-02-02 CN disclosed
US-10829485-B2 ATF6 inhibitors and uses thereof BLACK BELT TX LTD (GB) 2020-11-10 US disclosed
US-10829485-B2 ATF6 inhibitors and uses thereof BLACK BELT TX LTD (GB) 2020-11-10 US disclosed
EP-2390252-A1 New pyrazole derivatives Almirall, S.A. (ES) 2011-11-30 EP disclosed
EP-2390252-A1 New pyrazole derivatives Almirall, S.A. (ES) 2011-11-30 EP disclosed
WO-2011144338-A1 PYRAZOLE DERIVATIVES AS S1P1 AGONISTS ALMIRALL, S.A. (ES) 2011-11-24 WO disclosed
US-20110070297-A1 GLUCOKINASE ACTIVATORS TAKEDA SAN DIEGO, INC. (US) 2011-03-24 US disclosed
US-20110070297-A1 GLUCOKINASE ACTIVATORS TAKEDA SAN DIEGO, INC. (US) 2011-03-24 US disclosed
US-20070197532-A1 GLUCOKINASE ACTIVATORS TAKEDA SAN DIEGO, INC. 2007-08-23 US disclosed
US-20070197532-A1 GLUCOKINASE ACTIVATORS TAKEDA SAN DIEGO, INC. 2007-08-23 US disclosed
WO-2007061923-A2 GLUCOKINASE ACTIVATORS TAKEDA SAN DIEGO, INC. (US) 2007-05-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240124434-A1 ATF6 INHIBITORS AND USES THEREOF ATF4, XBP1, ATF1 NPC1 173/4885IDO1 4808/4885TDO2 4823/4885
US-12325702-B2 ATF6 inhibitors and uses thereof ATF4, XBP1, ATF1 NPC1 173/4885IDO1 4808/4885TDO2 4823/4885
US-10829485-B2 ATF6 inhibitors and uses thereof ATF4, XBP1, ATF1 NPC1 173/4885IDO1 4808/4885TDO2 4823/4885
US-20210221803-A1 ATF6 INHIBITORS AND USES THEREOF ATF4, XBP1, ATF1 NPC1 173/4885IDO1 4808/4885TDO2 4823/4885
US-20070197532-A1 GLUCOKINASE ACTIVATORS GCK, GCKR, GALK1 NPC1 2902/4885IDO1 4657/4885TDO2 3712/4885
US-20110070297-A1 GLUCOKINASE ACTIVATORS GCK, GCKR, GALK1 NPC1 2902/4885IDO1 4657/4885TDO2 3712/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.