SCHEMBL17397384

SCHEMBL17397384

COCCc1ccnc(N)n1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 4/20 0.44
CDK5R1 Q15078 4/20 0.44
CCNT1 O60563 3/20 0.44
CDK9 P50750 3/20 0.44
NUDT1 P36639 3/20 0.42
HRH4 Q9H3N8 4/20 0.40
HRH3 Q9Y5N1 4/20 0.39
DYRK1A Q13627 1/20 0.38
TLR8 Q9NR97 1/20 0.37
CCNA2 P20248 2/20 0.36
CDK2 P24941 2/20 0.36
CCNA1 P78396 2/20 0.36
AURKA O14965 1/20 0.35
HSP90AA1 P07900 1/20 0.35
PRKACA P17612 1/20 0.35
ADORA2A P29274 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6162470 0.81 NUDT1 (0.44) CDK5CDK5R1CCNT1CDK9NUDT1
SCHEMBL28128988 0.79 TSHR (0.35) CDK5CDK5R1CCNT1CDK9
SCHEMBL12336950 0.79 TLR8 (0.47) CDK5CDK5R1CCNT1CDK9NUDT1
SCHEMBL31298388 0.78 HRH4 (0.42) CDK5CDK5R1CCNT1CDK9NUDT1
SCHEMBL25942317 0.78 SMN1; SMN2 (0.38) CDK5CDK5R1CCNT1CDK9
SCHEMBL9324642 0.77 POLB (0.45) DYRK1AAURKAHSP90AA1PRKACAADORA2A
SCHEMBL12514073 0.76 TLR8 (0.53) NUDT1HRH4HRH3TLR8
SCHEMBL12439674 0.76 NUDT1 (0.51) NUDT1HRH4HRH3TLR8AURKA
SCHEMBL1016115 0.75 KCNH2 (0.54)
SCHEMBL8127847 0.75 HRH4 (0.42) NUDT1HRH4HRH3TLR8AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1109055-A 4-aminopyrimidine derivatives ONO PHARMACEUTICAL CO (JP) 1995-09-27 CN claimed
WO-2016000615-A1 HETEROARYL COMPOUNDS AND PHARMACEUTICAL APPLICATIONS THEREOF SUNSHINE LAKE PHARMA CO., LTD. (CN) 2016-01-07 WO disclosed
CN-1109055-A 4-aminopyrimidine derivatives ONO PHARMACEUTICAL CO (JP) 1995-09-27 CN disclosed