SCHEMBL1739916

SCHEMBL1739916

Cc1cc(COCCN2CCOCC2)nn1-c1csc2ccccc12

nearest known ligand 0.62

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 18/20 0.62
KCNH2 Q12809 1/20 0.46
HTR2B P41595 1/20 0.43
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
HIF1A Q16665 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1738636 0.88 SIGMAR1 (0.57) SIGMAR1HTR2BLMNA
SCHEMBL1740580 0.87 SIGMAR1 (0.58) SIGMAR1HTR2B
SCHEMBL1737439 0.77 SIGMAR1 (1.00) SIGMAR1KCNH2HTR2B
SCHEMBL1739361 0.74 SIGMAR1 (0.75) SIGMAR1KCNH2HTR2B
SCHEMBL9978613 0.73 SIGMAR1 (0.74) SIGMAR1KCNH2HTR2B
SCHEMBL1737898 0.73 SIGMAR1 (1.00) SIGMAR1KCNH2
SCHEMBL1738593 0.70 SIGMAR1 (0.46) SIGMAR1KCNH2ALDH1A1LMNA
SCHEMBL9978430 0.70 SIGMAR1 (0.68) SIGMAR1KCNH2
SCHEMBL9978406 0.68 SIGMAR1 (1.00) SIGMAR1KCNH2ALDH1A1
SCHEMBL1738639 0.68 SIGMAR1 (0.98) SIGMAR1KCNH2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2395003-A1 Pyrazole compounds as sigma receptor inhibitors Laboratorios Del. Dr. Esteve, S.A. (ES) 2011-12-14 EP claimed
EP-2395003-A1 Pyrazole compounds as sigma receptor inhibitors Laboratorios Del. Dr. Esteve, S.A. (ES) 2011-12-14 EP disclosed