SCHEMBL17405282

SCHEMBL17405282

c1ccc(-n2c(-c3ccc(-n4c5ccccc5c5c6c7ccccc7oc6c6c(c7ccccc7n6-c6ccccc6)c54)cc3)nc3ccccc32)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.47
ESR2 Q92731 1/20 0.47
GRIA1 P42261 1/20 0.44
CACNG8 Q8WXS5 1/20 0.44
CACNG2 Q9Y698 1/20 0.44
PTGS2 P35354 1/20 0.40
PRKACA P17612 1/20 0.39
RPS6KB1 P23443 1/20 0.39
GSK3B P49841 1/20 0.39
ROCK1 Q13464 1/20 0.39
HTT P42858 2/20 0.39
MAPK1 P28482 1/20 0.39
ALDH1A1 P00352 8/20 0.38
KMT2A Q03164 2/20 0.37
MEN1 O00255 1/20 0.37
HSP90AA1 P07900 1/20 0.37
MAPT P10636 1/20 0.37
RECQL P46063 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC8 Q9BY41 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17405297 0.98 ESR1 (0.50) ESR1ESR2GRIA1CACNG8CACNG2
SCHEMBL17405306 0.93 ESR1 (0.45) ESR1ESR2GRIA1CACNG8CACNG2
SCHEMBL17451684 0.93 ESR1 (0.46) ESR1ESR2GRIA1CACNG8CACNG2
SCHEMBL17405288 0.92 ESR1 (0.43) ESR1ESR2GRIA1CACNG8CACNG2
SCHEMBL17405293 0.92 ESR1 (0.43) ESR1ESR2GRIA1CACNG8CACNG2
SCHEMBL17405266 0.91 ALDH1A1 (0.44) ESR1ESR2HTTMAPK1ALDH1A1
SCHEMBL17405252 0.91 ESR1 (0.42) ESR1ESR2GRIA1CACNG8CACNG2
SCHEMBL17405285 0.88 MAPK1 (0.54) HTTMAPK1ALDH1A1KMT2AMEN1
SCHEMBL17405264 0.88 ALDH1A1 (0.47) PRKACARPS6KB1GSK3BROCK1HTT
SCHEMBL17405308 0.88 RECQL (0.43) ESR1ESR2PTGS2PRKACARPS6KB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9887367-B2 Heterocyclic compound, material for organic electroluminescent elements using same, organic electroluminescent element using same, and electronic device IDEMITSU KOSAN CO., LTD. (JP) 2018-02-06 US disclosed
US-9887367-B2 Heterocyclic compound, material for organic electroluminescent elements using same, organic electroluminescent element using same, and electronic device IDEMITSU KOSAN CO., LTD. (JP) 2018-02-06 US disclosed
US-20160005977-A1 HETEROCYCLIC COMPOUND, MATERIAL FOR ORGANIC ELECTROLUMINESCENT ELEMENTS USING SAME, ORGANIC ELECTROLUMINESCENT ELEMENT USING SAME, AND ELECTRONIC DEVICE IDEMITSU KOSAN CO., LTD. (JP) 2016-01-07 US disclosed
US-20160005977-A1 HETEROCYCLIC COMPOUND, MATERIAL FOR ORGANIC ELECTROLUMINESCENT ELEMENTS USING SAME, ORGANIC ELECTROLUMINESCENT ELEMENT USING SAME, AND ELECTRONIC DEVICE IDEMITSU KOSAN CO., LTD. (JP) 2016-01-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160005977-A1 HETEROCYCLIC COMPOUND, MATERIAL FOR ORGANIC ELECTROLUMINESCENT ELEMENTS USING SAME, ORGANIC ELECTROLUMINESCENT ELEMENT USING SAME, AND ELECTRONIC DEVICE ODC1, NOTUM, OR10J3 ESR1 29/4885ESR2 331/4885GRIA1 2263/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.