SCHEMBL1740722

SCHEMBL1740722

CCOC(=O)c1nn(CC)c(CC(C)C)c1Br

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.39
KMT2A Q03164 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
THRB P10828 1/20 0.39
HPGD P15428 1/20 0.39
PDE4B Q07343 6/20 0.38
PDE4A P27815 5/20 0.38
PDE4C Q08493 5/20 0.38
PDE4D Q08499 5/20 0.38
SMN1; SMN2 Q16637 3/20 0.36
MAPT P10636 3/20 0.36
MAPK1 P28482 2/20 0.36
ADORA3 P0DMS8 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
SLC5A1 P13866 1/20 0.35
SLC5A2 P31639 1/20 0.35
POLB P06746 1/20 0.35
NPC1 O15118 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1739254 0.86 ALDH1A1 (0.43) ALDH1A1KMT2AKDM4EMEN1THRB
SCHEMBL12181057 0.83 ALDH1A1 (0.42) ALDH1A1KMT2AKDM4EMEN1THRB
SCHEMBL1741283 0.82 NPC1 (0.39) ALDH1A1KDM4EMAPK1NPC1
SCHEMBL19618980 0.72 ALDH1A1 (0.39) ALDH1A1KMT2APDE4BPDE4APDE4C
SCHEMBL17478477 0.72 PDE4A (0.36) ALDH1A1KMT2AKDM4EMEN1HPGD
SCHEMBL19615264 0.72 ALDH1A1 (0.40) ALDH1A1KDM4EPDE4ASMN1; SMN2MAPT
SCHEMBL1739336 0.72 NPC1 (0.40) ALDH1A1KMT2AKDM4EMEN1THRB
SCHEMBL19615850 0.71 ALDH1A1 (0.39) ALDH1A1KDM4EPDE4ASMN1; SMN2MAPT
SCHEMBL19615364 0.70 NPC1 (0.36) ALDH1A1KDM4EHPGDPDE4BPDE4A
SCHEMBL19615438 0.70 SLC5A1 (0.42) ALDH1A1KDM4ESMN1; SMN2MAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2390252-A1 New pyrazole derivatives Almirall, S.A. (ES) 2011-11-30 EP disclosed
EP-2390252-A1 New pyrazole derivatives Almirall, S.A. (ES) 2011-11-30 EP disclosed