SCHEMBL17414533

SCHEMBL17414533

COc1cc(CO)cc(CC(=O)O)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.53
AKR1C3 P42330 1/20 0.53
AKR1C2 P52895 1/20 0.53
DAO P14920 1/20 0.47
RXRA P19793 2/20 0.46
RXRB P28702 1/20 0.46
RXRG P48443 1/20 0.46
TSHR P16473 2/20 0.45
HSD17B10 Q99714 2/20 0.45
ALOX15 P16050 1/20 0.45
KDM4E B2RXH2 2/20 0.45
POLB P06746 2/20 0.45
ABL1 P00519 1/20 0.45
MAPT P10636 1/20 0.45
RECQL P46063 1/20 0.45
RIN1 Q13671 1/20 0.45
CTDSP1 Q9GZU7 1/20 0.45
GAA P10253 2/20 0.45
ALDH1A1 P00352 1/20 0.45
NFKB1 P19838 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL347352 0.88 PTGS1 (0.59) PTGS1AKR1C3AKR1C2RXRARXRB
Hydrochloric Acid SCHEMBL2531690 0.86 PTGS1 (0.58) PTGS1AKR1C3AKR1C2RXRARXRB
SCHEMBL1621101 0.84 DAO (0.53) DAOMAPTALDH1A1CYP11B1CYP11B2
SCHEMBL31337475 0.84 PTGS1 (0.51) PTGS1AKR1C3AKR1C2RXRARXRB
SCHEMBL31337559 0.81 AKR1C2 (0.57) PTGS1AKR1C3AKR1C2RXRARXRB
SCHEMBL5315605 0.81 CALM1 (0.54) PTGS1AKR1C3AKR1C2RXRARXRB
SCHEMBL5742710 0.81 AKR1C2 (0.57) PTGS1AKR1C3AKR1C2RXRARXRB
SCHEMBL10350883 0.80 PTGS1 (0.51) PTGS1AKR1C3AKR1C2RXRARXRB
SCHEMBL6367068 0.80 PTGS1 (0.51) PTGS1AKR1C3AKR1C2RXRARXRB
SCHEMBL14856202 0.80 PTGS1 (0.51) PTGS1AKR1C3AKR1C2RXRARXRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170210728-A1 Cannabinergic Nitrate Esters And Related Analogs NORTHEASTERN UNIVERSITY 2017-07-27 US disclosed
US-9580400-B2 Cannabinergic nitrate esters and related analogs NORTHEASTERN UNIVERSITY (US) 2017-02-28 US disclosed
US-20160002195-A1 CANNABINERGIC NITRATE ESTERS AND RELATED ANALOGS NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2016-01-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160002195-A1 CANNABINERGIC NITRATE ESTERS AND RELATED ANALOGS CNR2, CNR1, CHRNB3 PTGS1 271/4885AKR1C3 1677/4885AKR1C2 1668/4885
US-20170210728-A1 Cannabinergic Nitrate Esters And Related Analogs CNR2, CNR1, CHRNB3 PTGS1 271/4885AKR1C3 1677/4885AKR1C2 1668/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.