SCHEMBL17425285

SCHEMBL17425285

O=C(NO)c1cnc(N2CC3[C@H]2CN3c2cccc(OC(F)I)c2)nc1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 20/20 0.40
HDAC1 Q13547 20/20 0.40
HDAC2 Q92769 20/20 0.40
HDAC6 Q9UBN7 20/20 0.40
HDAC4 P56524 17/20 0.40
HDAC7 Q8WUI4 17/20 0.40
HDAC10 Q969S8 17/20 0.40
HDAC11 Q96DB2 17/20 0.40
HDAC8 Q9BY41 17/20 0.40
HDAC9 Q9UKV0 17/20 0.40
HDAC5 Q9UQL6 17/20 0.40
CYP2D6 P10635 2/20 0.39
KCNH2 Q12809 1/20 0.39
CYP3A4 P08684 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16302041 0.92 ALOX15 (0.43) HDAC3HDAC1HDAC2HDAC6HDAC4
SCHEMBL16302012 0.85 HDAC1 (0.51) HDAC3HDAC1HDAC2HDAC6HDAC4
SCHEMBL16302010 0.84 HDAC6 (0.53) HDAC3HDAC1HDAC2HDAC6HDAC4
SCHEMBL16302045 0.83 HDAC1 (0.49) HDAC3HDAC1HDAC2HDAC6HDAC4
SCHEMBL8011347 0.83 HDAC1 (0.49) HDAC3HDAC1HDAC2HDAC6HDAC4
SCHEMBL16302069 0.81 HDAC6 (0.47) HDAC3HDAC1HDAC2HDAC6HDAC4
SCHEMBL16581065 0.81 HDAC6 (0.47) HDAC3HDAC1HDAC2HDAC6HDAC4
SCHEMBL16302008 0.80 HDAC1 (0.53) HDAC3HDAC1HDAC2HDAC6HDAC4
SCHEMBL16302006 0.80 HDAC6 (0.42) HDAC3HDAC1HDAC2HDAC6HDAC4
SCHEMBL18371376 0.80 HDAC6 (0.42) HDAC3HDAC1HDAC2HDAC6HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2966078-A2 Inhibitors of histone deacetylase MethylGene Inc. (CA) 2016-01-13 EP disclosed