SCHEMBL17425918

SCHEMBL17425918

FC(F)(F)Cn1cc(-c2ccc3c(n2)N(Cc2ccc4nccn4c2)NN3)cn1

nearest known ligand 0.59

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MET P08581 8/20 0.59
KEAP1 Q14145 1/20 0.34
LRRK2 Q5S007 2/20 0.34
PIM1 P11309 5/20 0.33
MERTK Q12866 1/20 0.31
NAMPT P43490 1/20 0.31
CYP1A2 P05177 1/20 0.31
METAP2 P50579 1/20 0.31
PIM3 Q86V86 4/20 0.31
PIM2 Q9P1W9 4/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21167810 0.88 MET (0.45) METKEAP1PIM1MERTK
SCHEMBL16882499 0.88 MET (0.64) METKEAP1LRRK2PIM1NAMPT
SCHEMBL21167627 0.87 MET (0.48) METKEAP1PIM1MERTKNAMPT
SCHEMBL12489788 0.78 MET (0.78) MET
SCHEMBL16882501 0.74 MET (0.54) METKEAP1NAMPT
SCHEMBL12487441 0.74 MET (1.00) MET
SCHEMBL21167805 0.73 MET (0.54) METKEAP1LRRK2NAMPT
SCHEMBL23128008 0.73 MET (0.46) METLRRK2PIM1PIM3PIM2
SCHEMBL22475811 0.72 MET (0.52) MET
SCHEMBL22475870 0.72 MET (0.53) METKEAP1LRRK2PIM1NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3511330-A1 SYNTHETIC INTERMEDIATE USEFUL IN THE PREPARATION OF TRIAZOLOPYRIDINE C-MET INHIBITORS Hutchison Medipharma Limited (CN) 2019-07-17 EP disclosed
EP-2966075-A1 CERTAIN TRIAZOLOPYRIDINES, COMPOSITIONS THEREOF AND THEIR USE IN THE TREATMENT OF CANCER. Hutchison Medipharma Limited (CN) 2016-01-13 EP disclosed