SCHEMBL1744238

SCHEMBL1744238

CC1Oc2cc[c]cc2N(C)C1=O

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 1/20 0.41
PDE3A Q14432 1/20 0.41
GRM4 Q14833 1/20 0.37
TSHR P16473 4/20 0.37
ALDH1A1 P00352 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
HTT P42858 1/20 0.37
MAOA P21397 1/20 0.36
ABCC8 Q09428 1/20 0.35
KCNJ11 Q14654 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
PARP1 P09874 1/20 0.33
THRB P10828 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2882448 0.80
SCHEMBL5799756 0.78 EGFR (0.33)
SCHEMBL3401752 0.78 TSHR (0.51) PDE3BPDE3ATSHRALDH1A1L3MBTL1
SCHEMBL29354025 0.78 TSHR (0.51) PDE3BPDE3ATSHRALDH1A1L3MBTL1
SCHEMBL10130347 0.72 TSHR (0.58) PDE3BPDE3AGRM4TSHRALDH1A1
SCHEMBL10129864 0.72 TSHR (0.58) PDE3BPDE3AGRM4TSHRALDH1A1
SCHEMBL10130351 0.72 TSHR (0.58) PDE3BPDE3AGRM4TSHRALDH1A1
SCHEMBL10129667 0.71 PDE3B (0.50) PDE3BPDE3AGRM4TSHRALDH1A1
SCHEMBL21475872 0.71 PDE3A (0.50) PDE3BPDE3AGRM4TSHRALDH1A1
SCHEMBL10129678 0.71 PDE3B (0.50) PDE3BPDE3AGRM4TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2385939-A1 DIHYDROPYRIDONE AMIDES AS P2X7 MODULATORS F. Hoffmann-La Roche AG (CH) 2011-11-16 EP disclosed
US-8041551-B1 Algorithm and architecture for multi-argument associative operations that minimizes the number of components using a latency of the components THE MATHWORKS, INC. (US) 2011-10-18 US disclosed
WO-2010072597-A1 DIHYDROPYRIDONE AMIDES AS P2X7 MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2010-07-01 WO disclosed