SCHEMBL3401752

SCHEMBL3401752

CC1Oc2ccccc2N(C)C1=O

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TSHR P16473 5/20 0.51
ALDH1A1 P00352 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
HTT P42858 1/20 0.51
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
PDE3B Q13370 1/20 0.46
PDE3A Q14432 1/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
MAOA P21397 1/20 0.44
PARP1 P09874 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29354025 1.00 TSHR (0.51) TSHRALDH1A1L3MBTL1HTTMEN1
SCHEMBL6114257 0.79 GABRP (0.42) TSHRALDH1A1L3MBTL1HTTKMT2A
2-Methyl-D-Diboa SCHEMBL13135829 0.79 ALDH1A1 (0.54) TSHRALDH1A1L3MBTL1HTTMEN1
SCHEMBL28045866 0.79 EGFR (0.41) TSHRALDH1A1L3MBTL1HTTMEN1
SCHEMBL18128200 0.79 TSHR (0.54) TSHRALDH1A1L3MBTL1HTTMEN1
SCHEMBL10130351 0.79 TSHR (0.58) TSHRALDH1A1MEN1KMT2APDE3B
SCHEMBL10130347 0.79 TSHR (0.58) TSHRALDH1A1MEN1KMT2APDE3B
SCHEMBL10129864 0.79 TSHR (0.58) TSHRALDH1A1MEN1KMT2APDE3B
SCHEMBL30036591 0.79 AADAT (0.41) TSHRALDH1A1L3MBTL1HTTMEN1
SCHEMBL1562017 0.79 AADAT (0.41) TSHRALDH1A1L3MBTL1HTTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019200202-A1 ANTAGONISTS OF HUMAN INTEGRIN (ALPHA4)(BETA7) MORPHIC THERAPEUTIC, INC. (US) 2019-10-17 WO disclosed
EP-2250169-A1 PYRIDO [4, 3-D]PYRIMIDINONE DERIVATIVES AS KINASE INHIBITORS IRM LLC (BM) 2010-11-17 EP disclosed
WO-2009099801-A1 PYRIDO [4, 3-D] PYRIMIDINONE DERIVATIVES AS KINASE INHIBITORS IRM LLC (BM) 2009-08-13 WO disclosed