SCHEMBL17469874

SCHEMBL17469874

CN(C)CCCNc1cc2cc(Br)ccc2cn1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 7/20 0.53
CLK4 Q9HAZ1 5/20 0.45
CDK5 Q00535 3/20 0.45
GSK3A P49840 1/20 0.45
CDK9 P50750 1/20 0.45
TAOK1 Q7L7X3 1/20 0.45
MAP4K4 O95819 4/20 0.44
MINK1 Q8N4C8 3/20 0.44
TYK2 P29597 2/20 0.44
SRPK1 Q96SB4 1/20 0.44
CLK2 P49760 4/20 0.43
DYRK1A Q13627 4/20 0.43
JAK2 O60674 3/20 0.43
GSK3B P49841 3/20 0.43
ROCK2 O75116 2/20 0.43
RPS6KB1 P23443 1/20 0.43
ROCK1 Q13464 1/20 0.43
FLT3 P36888 4/20 0.42
DNM2 P50570 2/20 0.41
DYRK3 O43781 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21512515 0.80 EGFR (0.50) EGFRMAPK1KDM4EALDH1A1
SCHEMBL29969091 0.80 EGFR (0.50) EGFRMAPK1KDM4EALDH1A1
SCHEMBL5495588 0.78 FLT3 (0.47) EGFRFLT3
SCHEMBL2621732 0.77 EGFR (0.49) EGFRFLT3MAPK1KDM4EALDH1A1
SCHEMBL12192994 0.73 IKBKB (0.46) DYRK1AGSK3BROCK1WNT1
SCHEMBL30834216 0.73 CYP1A2 (0.53) EGFRKDM4EALDH1A1
SCHEMBL27201452 0.73 CYP1A2 (0.53) EGFRKDM4EALDH1A1
SCHEMBL2671476 0.73 CLK4 (0.56) EGFRCLK4CDK5GSK3ACDK9
SCHEMBL26679803 0.72 ABL1 (0.46) CLK4CDK5GSK3ACDK9TAOK1
SCHEMBL1585465 0.72 EGFR (0.43) EGFRDNM2MAPK1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170174620-A1 LINKED DIARYL COMPOUNDS WITH ANTICANCER PROPERTIES AND METHODS OF USING THE SAME UNIVERSITY OF MARYLAND, COLLEGE PARK 2017-06-22 US disclosed
WO-2016014674-A1 LINKED DIARYL COMPOUNDS WITH ANTICANCER PROPERTIES AND METHODS OF USING THE SAME UNIVERSITY OF MARYLAND, COLLEGE PARK (US) 2016-01-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170174620-A1 LINKED DIARYL COMPOUNDS WITH ANTICANCER PROPERTIES AND METHODS OF USING THE SAME MCL1, DPYD, TOP2B EGFR 2900/4885CLK4 3290/4885CDK5 161/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.