SCHEMBL1748237

SCHEMBL1748237

COC(=O)[C@@H]1CCC[C@H]1C(=O)c1ccc(-c2ccc(Nc3nc4ccc(C)cc4o3)c(F)c2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 6/20 0.49
MAPT P10636 3/20 0.42
ALDH1A1 P00352 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
KDM4E B2RXH2 1/20 0.42
NPC1 O15118 1/20 0.42
HPGD P15428 1/20 0.42
NFKB1 P19838 1/20 0.42
RAB9A P51151 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
ATM Q13315 1/20 0.42
HSD17B10 Q99714 1/20 0.42
HCRTR1 O43613 2/20 0.37
AURKB Q96GD4 2/20 0.36
DYRK3 O43781 1/20 0.36
ROCK2 O75116 1/20 0.36
MAP4K4 O95819 1/20 0.36
ABL1 P00519 1/20 0.36
LCK P06239 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1748140 0.92 DGAT1 (0.58) DGAT1MAPTALDH1A1SMN1; SMN2KDM4E
SCHEMBL12315617 0.88 DGAT1 (0.46) DGAT1MAPTALDH1A1SMN1; SMN2KDM4E
SCHEMBL2308158 0.85 DGAT1 (0.56) DGAT1MAPTNPC1RAB9AAURKB
Bicarbonate SCHEMBL2311135 0.84 DGAT1 (0.44) DGAT1MAPTALDH1A1SMN1; SMN2KDM4E
SCHEMBL2311773 0.84 DGAT1 (0.61) DGAT1MAPTHCRTR1HDAC6
SCHEMBL2311873 0.84 DGAT1 (0.61) DGAT1MAPTHCRTR1HDAC6
SCHEMBL2311876 0.84 DGAT1 (0.61) DGAT1MAPTHCRTR1HDAC6
SCHEMBL2309693 0.83 DGAT1 (0.67) DGAT1HCRTR1
SCHEMBL2311010 0.81 DGAT1 (0.58) DGAT1MAPTRAB9A
SCHEMBL2307361 0.81 DGAT1 (0.58) DGAT1MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8013166-B2 Preparation and use of aryl alkyl acid derivatives for the treatment of obesity BAYER HEALTHCARE LLC (US) 2011-09-06 US disclosed
EP-1633722-B1 PREPARATION AND USE OF ARYL ALKYL ACID DERIVATIVES FOR THE TREATMENT OF OBESITY BAYER HEALTHCARE LLC (US) 2011-08-03 EP disclosed