SCHEMBL17484182

SCHEMBL17484182

CCc1nc2cc(C(F)(F)F)ccc2s1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.58
GAA P10253 1/20 0.58
MAPK1 P28482 1/20 0.58
RAB9A P51151 1/20 0.58
DYRK1A Q13627 1/20 0.52
AKR1B1 P15121 12/20 0.51
TRPV1 Q8NER1 2/20 0.48
ILK Q13418 2/20 0.47
AKR1A1 P14550 4/20 0.46
AKR1B10 O60218 1/20 0.45
GLO1 Q04760 1/20 0.45
ALOX5 P09917 1/20 0.44
EPHX2 P34913 1/20 0.44
SCN4A P35499 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20254213 0.88 DYRK1A (0.50) NPC1GAAMAPK1RAB9ADYRK1A
SCHEMBL10271381 0.87 EPHX2 (0.59) NPC1GAAMAPK1RAB9ADYRK1A
SCHEMBL14791428 0.85 NPC1 (0.59) NPC1GAAMAPK1RAB9ADYRK1A
SCHEMBL5632209 0.84 DYRK1A (0.50) DYRK1AAKR1B1TRPV1ILKAKR1A1
SCHEMBL359623 0.84 DYRK1A (0.49) DYRK1AAKR1B1TRPV1ILKAKR1A1
SCHEMBL360373 0.84 DYRK1A (0.49) DYRK1AAKR1B1TRPV1ILKAKR1A1
SCHEMBL3265720 0.84 LOXL2 (0.59) DYRK1AAKR1B1TRPV1ILKAKR1A1
SCHEMBL7082892 0.84 DYRK1A (0.49) DYRK1AAKR1B1TRPV1ILKAKR1A1
SCHEMBL20964606 0.83 DYRK1A (0.49) DYRK1AAKR1B1TRPV1ILKAKR1A1
Hydrochloric Acid SCHEMBL15708092 0.83 DYRK1A (0.48) DYRK1AAKR1B1TRPV1ILKAKR1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970158-B1 ALKYL-HETEROARYL SUBSTITUTED QUINONE DERIVATIVES FOR TREATMENT OF OXIDATIVE STRESS DISORDERS BIOELECTRON TECH CORP (US) 2019-02-20 EP disclosed
WO-2016019233-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE PHARMACYCLICS LLC (US) 2016-02-04 WO disclosed