SCHEMBL17485350

SCHEMBL17485350

Cc1nc2c(F)cc(-c3nc(Nc4ccc5[nH]cc(C6CCN(C)CC6)c5c4)ncc3F)cc2n1C(C)C

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 19/20 0.60
CDK1 P06493 14/20 0.60
CCNB1 P14635 11/20 0.60
CCNE1 P24864 10/20 0.60
CDK2 P24941 12/20 0.59
CDK6 Q00534 12/20 0.59
CDK9 P50750 6/20 0.59
CDK7 P50613 5/20 0.59
EGFR P00533 2/20 0.55
CCND3 P30281 3/20 0.53
CCNA2 P20248 2/20 0.53
KDR P35968 2/20 0.53
CCNT1 O60563 2/20 0.52
CHEK1 O14757 1/20 0.52
JAK2 O60674 1/20 0.52
CHEK2 O96017 1/20 0.52
RAF1 P04049 1/20 0.52
NTRK1 P04629 1/20 0.52
PDGFRB P09619 1/20 0.52
SRC P12931 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17485298 0.89 CDK4 (0.66) CDK4CDK1CCNB1CCNE1CDK2
SCHEMBL17477265 0.82 CDK4 (0.56) CDK4CDK1CCNB1CCNE1CDK2
SCHEMBL17477118 0.81 CDK4 (0.69) CDK4CDK1CCNB1CCNE1CDK2
SCHEMBL17489274 0.80 CDK4 (0.65) CDK4CDK1CCNB1CCNE1CDK2
SCHEMBL23010461 0.80 CDK4 (0.79) CDK4CDK2CDK6CDK9CDK7
SCHEMBL17488646 0.79 CDK4 (0.66) CDK4CDK1CCNB1CCNE1CDK2
SCHEMBL17488692 0.77 CDK4 (0.64) CDK4CDK1CCNB1CCNE1CDK2
SCHEMBL24333168 0.77 CDK4 (0.74) CDK4CDK1CCNB1CCNE1CDK2
SCHEMBL3447474 0.77 CDK4 (0.68) CDK4CDK1CCNB1CCNE1CDK2
SCHEMBL22172180 0.77 CDK4 (0.67) CDK4CDK1CCNB1CCNE1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016015604-A1 COMPOUNDS AS CDK SMALL-MOLECULE INHIBITORS AND USES THEREOF SUNSHINE LAKE PHARMA CO., LTD. (CN) 2016-02-04 WO disclosed