SCHEMBL17485372

SCHEMBL17485372

Cc1nc2c(F)cc(-c3nc(Nc4cc5c(cn4)CCNC5)ncc3F)cc2n1C(C)C

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 20/20 0.79
CDK6 Q00534 19/20 0.79
CDK2 P24941 18/20 0.79
CDK1 P06493 9/20 0.77
CDK7 P50613 7/20 0.77
CDK9 P50750 7/20 0.77
CDK5 Q00535 5/20 0.65
CCNB1 P14635 3/20 0.58
CCNE1 P24864 3/20 0.58
CIT O14578 1/20 0.58
GAK O14976 1/20 0.58
DYRK3 O43781 1/20 0.58
CCNT1 O60563 1/20 0.58
STK16 O75716 1/20 0.58
CCNK O75909 1/20 0.58
STK10 O94804 1/20 0.58
PRKD3 O94806 1/20 0.58
ABCB11 O95342 1/20 0.58
MAP4K4 O95819 1/20 0.58
CCNE2 O96020 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18288926 0.88 CDK4 (1.00) CDK4CDK6CDK2CDK1CDK7
Hydrochloric Acid SCHEMBL20548901 0.87 CDK4 (0.98) CDK4CDK6CDK2CDK1CDK7
SCHEMBL17485313 0.87 CDK4 (0.88) CDK4CDK6CDK2CDK1CDK7
SCHEMBL17477259 0.87 CDK4 (1.00) CDK4CDK6CDK2CDK1CDK7
SCHEMBL17477263 0.84 CDK4 (0.68) CDK4CDK6CDK2CDK1CDK7
SCHEMBL22003648 0.83 CDK4 (0.71) CDK4CDK6CDK2CDK1CDK7
SCHEMBL22003478 0.82 CDK4 (0.68) CDK4CDK6CDK2CDK1CDK7
SCHEMBL17485387 0.81 CDK4 (0.79) CDK4CDK6CDK2CDK1CDK7
SCHEMBL31066354 0.81 CDK4 (0.77) CDK4CDK6CDK2CDK1CDK7
SCHEMBL17489142 0.81 CDK4 (0.68) CDK4CDK6CDK2CDK1CDK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016015604-A1 COMPOUNDS AS CDK SMALL-MOLECULE INHIBITORS AND USES THEREOF SUNSHINE LAKE PHARMA CO., LTD. (CN) 2016-02-04 WO disclosed