SCHEMBL17488748

SCHEMBL17488748

Cc1nc2c(F)cc(-c3nc(Nc4ccc(CN5CCC(N6CCCCC6)CC5)cn4)ncc3F)cc2n1C(C)C

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 20/20 0.77
CDK1 P06493 16/20 0.77
CDK6 Q00534 13/20 0.77
CCND3 P30281 10/20 0.77
CCNE1 P24864 9/20 0.77
CCNB1 P14635 8/20 0.77
CDK2 P24941 5/20 0.77
CDK9 P50750 4/20 0.77
CCNA2 P20248 3/20 0.77
CCNT1 O60563 3/20 0.77
CDK7 P50613 3/20 0.77
CCNH P51946 2/20 0.77
CIT O14578 1/20 0.77
GAK O14976 1/20 0.77
DYRK3 O43781 1/20 0.77
STK16 O75716 1/20 0.77
CCNK O75909 1/20 0.77
STK10 O94804 1/20 0.77
PRKD3 O94806 1/20 0.77
ABCB11 O95342 1/20 0.77

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17477131 0.99 CDK4 (0.78) CDK4CDK1CDK6CCND3CCNE1
SCHEMBL17488966 0.94 CDK4 (0.76) CDK4CDK1CDK6CCND3CCNE1
SCHEMBL17489052 0.93 CDK4 (0.88) CDK4CDK1CDK6CCND3CCNE1
SCHEMBL17488745 0.93 CDK4 (0.88) CDK4CDK1CDK6CCND3CCNE1
SCHEMBL21658739 0.93 CDK4 (0.87) CDK4CDK1CDK6CCND3CCNE1
SCHEMBL17488760 0.92 CDK4 (0.88) CDK4CDK1CDK6CCND3CCNE1
SCHEMBL17489051 0.92 CDK4 (0.73) CDK4CDK1CDK6CCND3CCNE1
SCHEMBL17488700 0.90 CDK4 (0.82) CDK4CDK1CDK6CCND3CCNE1
SCHEMBL26296402 0.89 CDK4 (0.83) CDK4CDK1CDK6CCND3CCNE1
SCHEMBL17488797 0.89 CDK4 (0.80) CDK4CDK1CDK6CCND3CCNE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016015605-A1 COMPOUNDS AS CDK SMALL-MOLECULE INHIBITORS AND USES THEREOF SUNSHINE LAKE PHARMA CO., LTD. (CN) 2016-02-04 WO disclosed