SCHEMBL17489331

SCHEMBL17489331

C#Cc1cc(C(C)C)ccc1OCc1cccc(F)c1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.47
ERBB2 P04626 1/20 0.47
MAOB P27338 9/20 0.44
MAOA P21397 2/20 0.43
MRGPRX4 Q96LA9 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
MAPT P10636 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
IDO1 P14902 1/20 0.40
AGXT P21549 1/20 0.40
LMNA P02545 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
FFAR1 O14842 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11949601 0.83 EGFR (0.49) EGFRERBB2MAOBMAOAMRGPRX4
SCHEMBL6960989 0.82 EGFR (0.52) EGFRERBB2MAOBMAOAMAPT
SCHEMBL13900992 0.81 EGFR (0.53) EGFRERBB2MAOBMRGPRX4
SCHEMBL4028363 0.81 MAOB (0.57) EGFRERBB2MAOBMAOACYP1A2
SCHEMBL15701549 0.80 EGFR (0.47) EGFRERBB2MAOBMAOAMRGPRX4
SCHEMBL24726468 0.79 MAOB (0.48) MAOBMRGPRX4IDO1AGXTLMNA
SCHEMBL24726471 0.76 MAOB (0.69) MAOBMAOAMRGPRX4FFAR1
SCHEMBL18253179 0.74 MAOB (0.66) MAOBMAOAMRGPRX4
SCHEMBL14200028 0.72 MAOB (0.56) MAOB
SCHEMBL20004351 0.71 IDO1 (0.50) MAOBMAOAMRGPRX4IDO1AGXT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160031860-A1 ALKYNE SUBSTITUTED QUINAZOLINE COMPOUND AND METHODS OF USE NEWGEN THERAPEUTICS INC (US) 2016-02-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160031860-A1 ALKYNE SUBSTITUTED QUINAZOLINE COMPOUND AND METHODS OF USE ERBB2, ERBB4, ERBB3 EGFR 5/4885ERBB2 1/4885MAOB 2081/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.