SCHEMBL17505000

SCHEMBL17505000

CC(C)(O)[C@@H]1CN(c2cccc(S(C)(=O)=O)c2)CCN1C(=O)O

nearest known ligand 0.77

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 19/20 0.77
NR1H3 Q13133 16/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17519220 0.87 NR1H2 (1.00) NR1H2NR1H3
SCHEMBL21442550 0.87 NR1H2 (1.00) NR1H2NR1H3
SCHEMBL21433374 0.82 NR1H2 (0.60) NR1H2NR1H3
SCHEMBL21433371 0.82 NR1H2 (0.60) NR1H2NR1H3
SCHEMBL21433339 0.81 NR1H2 (0.74) NR1H2NR1H3
SCHEMBL21433337 0.81 NR1H2 (0.74) NR1H2NR1H3
SCHEMBL2224887 0.75 NR1H2 (0.45) NR1H2NR1H3
SCHEMBL29252729 0.75 AGTR2 (0.48) NR1H2NR1H3
SCHEMBL673259 0.74 NR1H2 (0.51) NR1H2NR1H3
SCHEMBL11963285 0.74 NR1H2 (0.44) NR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3177617-A1 PIPERAZINE DERIVATIVES AS LIVER X RECEPTOR MODULATORS Vitae Pharmaceuticals, Inc. (US) 2017-06-14 EP disclosed
WO-2016022521-A1 PIPERAZINE DERIVATIVES AS LIVER X RECEPTOR MODULATORS VITAE PHARMACEUTICALS, INC. (US) 2016-02-11 WO disclosed