SCHEMBL17508159

SCHEMBL17508159

Cc1ccc(-c2ccc(C=O)cc2)c(F)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.52
HDAC1 Q13547 3/20 0.45
KDM1A O60341 2/20 0.45
HDAC6 Q9UBN7 2/20 0.45
KIF11 P52732 1/20 0.44
NFE2L2 Q16236 3/20 0.42
PTGS1 P23219 2/20 0.41
PTGS2 P35354 2/20 0.40
PDE3B Q13370 1/20 0.40
PDE3A Q14432 1/20 0.40
AKR1C3 P42330 1/20 0.40
AKR1C2 P52895 1/20 0.40
HDAC2 Q92769 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
DRD1 P21728 3/20 0.39
DRD2 P14416 1/20 0.38
DRD4 P21917 1/20 0.38
DRD5 P21918 1/20 0.38
DRD3 P35462 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21386564 0.91 CYP2A6 (0.55) CYP2A6HDAC1KDM1AHDAC6KIF11
SCHEMBL17408975 0.86 CYP2A6 (0.52) CYP2A6KIF11NFE2L2PTGS1PTGS2
SCHEMBL13967517 0.84 PTGS2 (0.46) HDAC1KDM1AHDAC6NFE2L2PTGS1
SCHEMBL10018702 0.82 PTGS2 (0.48) HDAC1KDM1AHDAC6NFE2L2PTGS1
SCHEMBL21093877 0.82 HDAC1 (0.42) HDAC1KDM1AHDAC6NFE2L2PTGS1
SCHEMBL2012266 0.81 CYP2A6 (0.56) CYP2A6PTGS1AKR1C3AKR1C2DRD1
SCHEMBL416643 0.81 PTGS1 (0.51) KIF11NFE2L2PTGS1PTGS2DRD1
SCHEMBL31120808 0.81 PTGS1 (0.51) KIF11NFE2L2PTGS1PTGS2DRD1
SCHEMBL10013948 0.81 PTGS2 (0.47) HDAC1KDM1AHDAC6NFE2L2PTGS1
SCHEMBL7791196 0.79 NPC1 (0.57) HDAC1KDM1AHDAC6NFE2L2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016019588-A1 OXACAZONE COMPOUNDS TO TREAT CLOSTRIDIUM DIFFICILE THE BROAD INSTITUTE, INC. (US) 2016-02-11 WO disclosed
WO-2016019588-A1 OXACAZONE COMPOUNDS TO TREAT CLOSTRIDIUM DIFFICILE THE BROAD INSTITUTE, INC. (US) 2016-02-11 WO disclosed