SCHEMBL17529341

SCHEMBL17529341

CN(CCN1CCOCC1)C(=O)c1cccc(C(=O)O)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 1/20 0.43
TACR3 P29371 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
KMT2A Q03164 4/20 0.42
ALDH1A1 P00352 2/20 0.42
MAPT P10636 2/20 0.42
MEN1 O00255 2/20 0.42
KDM4E B2RXH2 1/20 0.41
ALOX15 P16050 1/20 0.41
TSHR P16473 1/20 0.41
ACMSD Q8TDX5 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
PIK3CD O00329 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CHRM3 P20309 1/20 0.41
GNE Q9Y223 1/20 0.41
HRH3 Q9Y5N1 1/20 0.40
OPRM1 P35372 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28037481 0.79 ALDH1A1 (0.58) TACR1TACR3KMT2AALDH1A1MAPT
SCHEMBL40396 0.79 CASR (0.51) TACR1TACR3KMT2AALDH1A1MAPT
SCHEMBL29289842 0.76 KDM4E (0.55) KMT2AMEN1KDM4EALOX15TSHR
SCHEMBL16691265 0.73 PIK3CD (0.43) TACR1TACR3KMT2AALDH1A1MAPT
SCHEMBL40051 0.73 DRD4 (0.53) TACR1TACR3KMT2AALDH1A1MAPT
SCHEMBL12505784 0.73 DRD4 (0.50) TACR1TACR3KMT2AALDH1A1MAPT
SCHEMBL28280909 0.72 ALDH1A1 (0.50) TACR1TACR3NPSR1KMT2AALDH1A1
SCHEMBL28628270 0.72 KDM4E (0.59) KMT2AALDH1A1MAPTMEN1KDM4E
SCHEMBL31679380 0.72 CXCR4 (0.69) KMT2AALDH1A1MAPTMEN1KDM4E
SCHEMBL465725 0.72 CXCR4 (0.69) KMT2AALDH1A1MAPTMEN1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105658635-B Thieno naphthenic base or thieno heterocycle analog derivative, preparation method and its application in medicine 江苏恒瑞医药股份有限公司 2019-03-08 CN disclosed
WO-2016026372-A1 THIENOCYCLOALKYL OR THIENOHETEROCYCLIC DERIVATIVES, PREPARATION METHOD THEREOF AND USE THEREOF IN MEDICINE 江苏恒瑞医药股份有限公司 2016-02-25 WO disclosed