SCHEMBL17533535

SCHEMBL17533535

COC(=O)C(CCC(=O)O)CP(=O)(O)O

nearest known ligand 0.65

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
FOLH1 Q04609 9/20 0.65
NAALAD2 Q9Y3Q0 1/20 0.65
GRM3 Q14832 2/20 0.50
GGH Q92820 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19225283 0.86 FOLH1 (0.47) FOLH1NAALAD2GRM3GGH
SCHEMBL19220645 0.86 FOLH1 (0.46) FOLH1NAALAD2GRM3
SCHEMBL17504780 0.86 FOLH1 (0.46) FOLH1NAALAD2GRM3
SCHEMBL5134136 0.85 GRM3 (0.74) FOLH1NAALAD2GRM3
SCHEMBL16528808 0.79 FOLH1 (1.00) FOLH1NAALAD2GRM3
SCHEMBL383173 0.79 FOLH1 (1.00) FOLH1NAALAD2GRM3
SCHEMBL16528703 0.79 FOLH1 (1.00) FOLH1NAALAD2GRM3
SCHEMBL19225240 0.78 FOLH1 (0.54) FOLH1NAALAD2GRM3
SCHEMBL5134133 0.78 GRM3 (0.68) FOLH1NAALAD2GRM3
SCHEMBL19242717 0.78 FOLH1 (0.54) FOLH1NAALAD2GRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11325931-B2 Prodrugs of prostate specific membrane antigen (PSMA) inhibitor THE JOHNS HOPKINS UNIVERSITY (US) 2022-05-10 US disclosed
US-20200399298-A1 PRODRUGS OF PROSTATE SPECIFIC MEMBRANE ANTIGEN (PSMA) INHIBITOR THE JOHNS HOPKINS UNIVERSITY 2020-12-24 US disclosed
US-20200069706-A1 PRODRUGS OF 2-PMPA FOR HEALTHY TISSUE PROTECTION DURING PSMA-TARGETED CANCER IMAGING OR RADIOTHERAPY BAYER HEALTHCARE HOLDINGS LLC 2020-03-05 US disclosed
US-10544176-B2 Prodrugs of prostate specific membrane antigen (PSMA) inhibitor THE JOHNS HOPKINS UNIVERSITY (US) 2020-01-28 US disclosed
US-9988407-B2 Prodrugs of prostate specific membrane antigen (PSMA) inhibitor THE JOHNS HOPKINS UNIVERSITY (US) 2018-06-05 US disclosed
US-9988407-B2 Prodrugs of prostate specific membrane antigen (PSMA) inhibitor THE JOHNS HOPKINS UNIVERSITY (US) 2018-06-05 US disclosed
US-20170226141-A1 PRODRUGS OF PROSTATE SPECIFIC MEMBRANE ANTIGEN (PSMA) INHIBITOR THE JOHNS HOPKINS UNIVERSITY (US) 2017-08-10 US disclosed
US-20170226141-A1 PRODRUGS OF PROSTATE SPECIFIC MEMBRANE ANTIGEN (PSMA) INHIBITOR THE JOHNS HOPKINS UNIVERSITY (US) 2017-08-10 US disclosed
WO-2016022827-A1 PRODRUGS OF PROSTATE SPECIFIC MEMBRANE ANTIGEN (PSMA) INHIBITOR THE JOHNS HOPKINS UNIVERSITY (US) 2016-02-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11325931-B2 Prodrugs of prostate specific membrane antigen (PSMA) inhibitor FOLH1, KLK3, DNPEP FOLH1 1/4885NAALAD2 111/4885GRM3 1812/4885
US-20170226141-A1 PRODRUGS OF PROSTATE SPECIFIC MEMBRANE ANTIGEN (PSMA) INHIBITOR FOLH1, KLK3, DNPEP FOLH1 1/4885NAALAD2 111/4885GRM3 1812/4885
US-20200399298-A1 PRODRUGS OF PROSTATE SPECIFIC MEMBRANE ANTIGEN (PSMA) INHIBITOR FOLH1, KLK3, DNPEP FOLH1 1/4885NAALAD2 89/4885GRM3 1678/4885
US-20200069706-A1 PRODRUGS OF 2-PMPA FOR HEALTHY TISSUE PROTECTION DURING PSMA-TARGETED CANCER IMAGING OR RADIOTHERAPY PLPBP, PTMA, PTPA FOLH1 19/4885NAALAD2 406/4885GRM3 3112/4885
US-10544176-B2 Prodrugs of prostate specific membrane antigen (PSMA) inhibitor FOLH1, KLK3, DNPEP FOLH1 1/4885NAALAD2 111/4885GRM3 1812/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.