SCHEMBL1753773

SCHEMBL1753773

O=C(O)COc1ccc(Cl)cc1-c1ccc(C(=O)O)cc1

nearest known ligand 0.76

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 13/20 0.76
PTGER1 P34995 1/20 0.62
TDP1 Q9NUW8 2/20 0.59
MAPT P10636 1/20 0.58
TSHR P16473 1/20 0.54
SRD5A2 P31213 1/20 0.51
MRGPRX4 Q96LA9 1/20 0.51
PTGDR Q13258 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1753654 0.91 PTGDR2 (0.85) PTGDR2TDP1MAPTTSHRPTGDR
SCHEMBL12147097 0.87 PTGDR2 (1.00) PTGDR2TDP1MAPTTSHR
SCHEMBL16199771 0.87 PTGDR2 (0.58) PTGDR2PTGER1TDP1MAPTTSHR
SCHEMBL12147241 0.85 PTGDR2 (0.67) PTGDR2PTGER1TDP1MAPTTSHR
SCHEMBL1753406 0.83 PTGDR2 (0.72) PTGDR2TDP1MAPTTSHR
SCHEMBL12147488 0.83 PTGDR2 (0.76) PTGDR2TDP1MAPTTSHRPTGDR
SCHEMBL1753771 0.82 PTGDR2 (0.76) PTGDR2TDP1MAPTTSHR
SCHEMBL1753551 0.81 PTGDR2 (0.71) PTGDR2TDP1MAPTTSHR
SCHEMBL1753560 0.81 PTGDR2 (0.80) PTGDR2
SCHEMBL12147409 0.81 PTGDR2 (0.69) PTGDR2PTGER1TDP1MAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8158820-B2 Compounds ASTRAZENECA AB (SE) 2012-04-17 US claimed
US-20110166117-A1 Novel Compounds ASTRAZENECA AB (SE) 2011-07-07 US claimed
EP-1611091-B1 Substituted phenylalkanoic acid derivatives and their use for respiratory disease treatment ASTRAZENECA AB (SE) 2014-10-29 EP disclosed
US-8158820-B2 Compounds ASTRAZENECA AB (SE) 2012-04-17 US disclosed
US-8158820-B2 Compounds ASTRAZENECA AB (SE) 2012-04-17 US disclosed
US-8158820-B2 Compounds ASTRAZENECA AB (SE) 2012-04-17 US disclosed
US-20110166117-A1 Novel Compounds ASTRAZENECA AB (SE) 2011-07-07 US disclosed
US-20110166117-A1 Novel Compounds ASTRAZENECA AB (SE) 2011-07-07 US disclosed
US-20110166117-A1 Novel Compounds ASTRAZENECA AB (SE) 2011-07-07 US disclosed
US-20060264435-A1 Novel compounds ASTRAZENECA AB (SE) 2006-11-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110166117-A1 Novel Compounds ADRA2C, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, HCAR2 PTGDR2 438/4885PTGER1 351/4885TDP1 3990/4885
US-20060264435-A1 Novel compounds ADRA2C, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, HCAR2 PTGDR2 438/4885PTGER1 351/4885TDP1 3990/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.