SCHEMBL17538367

SCHEMBL17538367

CCN1CCN(c2nccc(C(F)(F)F)n2)C[C@H]1C

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 1/20 0.51
CHRM2 P08172 1/20 0.47
CHRM3 P20309 1/20 0.47
RBP4 P02753 1/20 0.46
HTR2C P28335 5/20 0.45
HTR2A P28223 4/20 0.45
HTR2B P41595 4/20 0.45
KDM4E B2RXH2 2/20 0.44
OGA O60502 1/20 0.44
PKM P14618 1/20 0.42
KMT2A Q03164 1/20 0.42
SLC6A7 Q99884 1/20 0.42
NR1H3 Q13133 3/20 0.41
NR1H2 P55055 2/20 0.41
GPBAR1 Q8TDU6 1/20 0.41
ALDH1A1 P00352 1/20 0.41
ACACB O00763 1/20 0.41
PARP1 P09874 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17538377 1.00 ADRB1 (0.51) ADRB1CHRM2CHRM3RBP4HTR2C
SCHEMBL12153215 0.88 ADRB1 (0.47) ADRB1CHRM2CHRM3RBP4HTR2C
SCHEMBL13677241 0.83 ADRB1 (0.55) ADRB1CHRM2CHRM3RBP4HTR2C
SCHEMBL13677250 0.83 ADRB1 (0.55) ADRB1CHRM2CHRM3RBP4HTR2C
SCHEMBL12153149 0.80 ADRB1 (0.51) ADRB1CHRM2CHRM3RBP4HTR2C
SCHEMBL13676971 0.80 ADRB1 (0.51) ADRB1CHRM2CHRM3RBP4HTR2C
SCHEMBL19035671 0.78 GRM1 (0.46) KDM4ESLC6A7
SCHEMBL8354208 0.78 ADRB1 (0.78) ADRB1RBP4HTR2CHTR2AHTR2B
SCHEMBL13059864 0.76 ADRB1 (0.55) ADRB1RBP4HTR2CHTR2AHTR2B
SCHEMBL1735009 0.75 ADRB1 (0.66) ADRB1RBP4HTR2CHTR2AHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1954287-B2 CETP INHIBITORS MERCK SHARP & DOHME (US) 2016-02-24 EP disclosed