SCHEMBL17539710

SCHEMBL17539710

ICCc1ccc(Nc2ncc(-c3cccnc3)s2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 13/20 0.60
NAMPT P43490 1/20 0.48
HDAC3 O15379 5/20 0.47
ABL1 P00519 5/20 0.47
PDGFRB P09619 5/20 0.47
HDAC4 P56524 5/20 0.47
HDAC1 Q13547 5/20 0.47
HDAC7 Q8WUI4 5/20 0.47
HDAC2 Q92769 5/20 0.47
HDAC10 Q969S8 5/20 0.47
HDAC11 Q96DB2 5/20 0.47
HDAC8 Q9BY41 5/20 0.47
HDAC6 Q9UBN7 5/20 0.47
HDAC9 Q9UKV0 5/20 0.47
HDAC5 Q9UQL6 5/20 0.47
MEN1 O00255 2/20 0.45
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
KMT2A Q03164 2/20 0.45
KIT P10721 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17539705 0.80 KDR (0.55) KDRNAMPTHDAC3ABL1PDGFRB
Bromide SCHEMBL29350593 0.79 KDR (0.54) KDRNAMPTHDAC3ABL1PDGFRB
SCHEMBL22560265 0.75 KDR (0.73) KDRNAMPTHDAC3ABL1PDGFRB
SCHEMBL6330184 0.75 KDR (1.00) KDRHDAC3ABL1PDGFRBHDAC4
SCHEMBL6330404 0.72 KDR (1.00) KDRNAMPTROCK1
SCHEMBL24225743 0.72 KDR (0.40) KDRNAMPTHDAC3ABL1PDGFRB
SCHEMBL13701560 0.71 KDR (0.81) KDRNPC1RAB9A
SCHEMBL12909537 0.71 KDR (0.59) KDRHDAC3ABL1PDGFRBHDAC4
SCHEMBL3651635 0.71 KDR (1.00) KDRNAMPTROCK1
SCHEMBL12890440 0.69 KDR (0.56) KDRHDAC3ABL1PDGFRBHDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016028325-A1 TRPA1 AND TRPV4 INHIBITORS AND METHODS OF USING THE SAME FOR ORGAN-SPECIFIC INFLAMMATION AND ITCH DUKE UNIVERSITY (US) 2016-02-25 WO disclosed