SCHEMBL1754669

SCHEMBL1754669

COc1c(OCc2ccc(C(C)=O)cc2)cccc1C1SC(c2ccc(F)cc2)=NN1C(=O)c1ccc(C(F)(F)F)cc1C(F)(F)F

nearest known ligand 0.56

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 19/20 0.56
NR1H3 Q13133 14/20 0.55
RXRA P19793 1/20 0.38
RXRB P28702 1/20 0.38
RXRG P48443 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1754489 0.94 NR1H2 (0.56) NR1H2NR1H3RXRARXRBRXRG
SCHEMBL1754655 0.85 NR1H2 (0.59) NR1H2NR1H3
SCHEMBL1754023 0.84 NR1H2 (0.59) NR1H2NR1H3
SCHEMBL13576036 0.81 RXRA (0.39) RXRARXRBRXRG
SCHEMBL1754700 0.80 NR1H2 (0.59) NR1H2NR1H3
SCHEMBL1754689 0.80 NR1H2 (0.59) NR1H2NR1H3
SCHEMBL1754638 0.80 NR1H2 (0.65) NR1H2NR1H3
SCHEMBL1754344 0.79 NR1H2 (0.59) NR1H2NR1H3RXRA
SCHEMBL1754027 0.79 NR1H2 (0.78) NR1H2NR1H3
SCHEMBL1754682 0.79 NR1H2 (0.67) NR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8158662-B2 Compounds and compositions as LXR modulators HAMILTON (BM) 2012-04-17 US disclosed