SCHEMBL1754671

SCHEMBL1754671

COc1c(OCc2ccc(S(C)(=O)=O)cc2)cccc1C1SC(c2ccc(F)cc2)=NN1C(=O)c1ccccc1C

nearest known ligand 0.63

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 18/20 0.63
NR1H3 Q13133 14/20 0.63
PTGS2 P35354 1/20 0.42
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1754372 0.93 NR1H2 (0.62) NR1H2NR1H3MEN1KMT2A
SCHEMBL1754614 0.93 NR1H2 (0.57) NR1H2NR1H3PTGS2KMT2A
SCHEMBL1753970 0.87 NR1H2 (0.57) NR1H2NR1H3KMT2A
SCHEMBL1754672 0.85 NR1H2 (0.53) NR1H2NR1H3PTGS2
SCHEMBL1754022 0.85 NR1H2 (0.65) NR1H2NR1H3
SCHEMBL1754638 0.85 NR1H2 (0.65) NR1H2NR1H3MEN1KMT2A
SCHEMBL11997940 0.85 NR1H2 (0.71) NR1H2NR1H3MEN1KMT2A
SCHEMBL1753956 0.85 NR1H2 (0.64) NR1H2NR1H3MEN1KMT2A
SCHEMBL1753883 0.85 NR1H2 (0.62) NR1H2NR1H3MEN1KMT2A
SCHEMBL1754667 0.84 NR1H2 (0.70) NR1H2NR1H3MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8158662-B2 Compounds and compositions as LXR modulators HAMILTON (BM) 2012-04-17 US disclosed