SCHEMBL17547019

SCHEMBL17547019

COc1ccc(-c2cccc(I)c2)cn1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 2/20 0.65
HSD17B2 P37059 2/20 0.65
ADORA2A P29274 1/20 0.50
ADORA1 P30542 1/20 0.50
CYP2A6 P11509 2/20 0.49
PDGFRB P09619 1/20 0.48
PDGFRA P16234 1/20 0.48
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
KDR P35968 3/20 0.47
PIK3CA P42336 2/20 0.47
PIK3CD O00329 1/20 0.47
PIP5K1C O60331 1/20 0.47
PIK3CB P42338 1/20 0.47
PI4KA P42356 1/20 0.47
PIK3CG P48736 1/20 0.47
PI4KB Q9UBF8 1/20 0.47
MKNK1 Q9BUB5 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12498936 0.81 HSD17B1 (0.67) HSD17B1HSD17B2ADORA2AADORA1CYP2A6
SCHEMBL13575386 0.81 HSD17B1 (0.67) HSD17B1HSD17B2ADORA2AADORA1CYP2A6
SCHEMBL13575381 0.81 HSD17B1 (0.67) HSD17B1HSD17B2ADORA2AADORA1CYP2A6
SCHEMBL17742850 0.80 MKNK1 (0.57) HSD17B1HSD17B2CYP2A6PDGFRBPDGFRA
SCHEMBL980158 0.80 HSD17B1 (0.65) HSD17B1HSD17B2ADORA2AADORA1CYP2A6
SCHEMBL5673332 0.80 HSD17B1 (0.97) HSD17B1HSD17B2ADORA2AADORA1CYP2A6
SCHEMBL13575397 0.80 HSD17B1 (0.65) HSD17B1HSD17B2ADORA2AADORA1CYP2A6
SCHEMBL31174412 0.80 CYP2A6 (0.68) HSD17B1HSD17B2CYP2A6PDGFRBPDGFRA
SCHEMBL3754419 0.80 CYP2A6 (0.68) HSD17B1HSD17B2CYP2A6PDGFRBPDGFRA
SCHEMBL5714627 0.79 HSD17B1 (0.63) HSD17B1HSD17B2ADORA2AADORA1CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3070081-A1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION Gilead Sciences, Inc. (US) 2016-09-21 EP disclosed
EP-2788336-B1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES INC (US) 2016-03-02 EP disclosed