SCHEMBL17553471

SCHEMBL17553471

C=CC(=O)Nc1cc(Nc2nccc(-c3cn(CCO)c4ccccc34)n2)c(OC)cc1N(C)CCN(C)C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 20/20 1.00
MLNR O43193 1/20 0.85
KDM1A O60341 1/20 0.85
ABCB11 O95342 1/20 0.85
ERBB2 P04626 1/20 0.85
INSR P06213 1/20 0.85
CHRM2 P08172 1/20 0.85
HTR1A P08908 1/20 0.85
ADORA3 P0DMS8 1/20 0.85
DRD2 P14416 1/20 0.85
NQO2 P16083 1/20 0.85
ADRA2C P18825 1/20 0.85
DRD1 P21728 1/20 0.85
ERBB3 P21860 1/20 0.85
SLC6A2 P23975 1/20 0.85
HTR2A P28223 1/20 0.85
HTR2C P28335 1/20 0.85
ADORA2A P29274 1/20 0.85
SLC6A4 P31645 1/20 0.85
CCKAR P32238 1/20 0.85

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22968448 0.95 EGFR (0.90) EGFRMLNRKDM1AABCB11ERBB2
SCHEMBL28409356 0.94 EGFR (0.91) EGFRMLNRKDM1AABCB11ERBB2
SCHEMBL24117622 0.94 EGFR (0.90) EGFRMLNRKDM1AABCB11ERBB2
SCHEMBL17683310 0.94 EGFR (1.00) EGFRMLNRKDM1AABCB11ERBB2
SCHEMBL28412579 0.93 EGFR (0.91) EGFRMLNRKDM1AABCB11ERBB2
SCHEMBL17553693 0.93 EGFR (0.91) EGFRMLNRKDM1AABCB11ERBB2
SCHEMBL17683234 0.92 EGFR (0.85) EGFRMLNRKDM1AABCB11ERBB2
SCHEMBL17683083 0.92 EGFR (0.85) EGFRMLNRKDM1AABCB11ERBB2
SCHEMBL28409189 0.92 EGFR (0.86) EGFRMLNRKDM1AABCB11ERBB2
Osimertinib SCHEMBL14660911 0.92 EGFR (1.00) EGFRMLNRKDM1AABCB11ERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113121575-A (substituted phenyl) (substituted pyrimidine) amino derivative and preparation method and pharmaceutical application thereof 四川海思科制药有限公司 2021-07-16 CN disclosed
CN-106458969-A (substituted phenyl) (substituted pyrimidine) amino derivative and preparation method and pharmaceutical application thereof 四川海思科制药有限公司 2017-02-22 CN disclosed
WO-2016029839-A1 (SUBSTITUTED PHENYL) (SUBSTITUTED PYRIMIDINE) AMINO DERIVATIVE, PREPARATION METHOD THEREFOR, AND MEDICATION USE 四川海思科制药有限公司 2016-03-03 WO disclosed