SCHEMBL28409356

SCHEMBL28409356

C=CC(=O)Nc1cc(Nc2nccc(-c3cn(CO)c4ccccc34)n2)c(OC)cc1N(C)CCN(C)C

nearest known ligand 0.91

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 20/20 0.91
KCNH2 Q12809 2/20 0.84
MLNR O43193 1/20 0.84
KDM1A O60341 1/20 0.84
ABCB11 O95342 1/20 0.84
ERBB2 P04626 1/20 0.84
INSR P06213 1/20 0.84
CHRM2 P08172 1/20 0.84
HTR1A P08908 1/20 0.84
ADORA3 P0DMS8 1/20 0.84
DRD2 P14416 1/20 0.84
NQO2 P16083 1/20 0.84
ADRA2C P18825 1/20 0.84
DRD1 P21728 1/20 0.84
ERBB3 P21860 1/20 0.84
SLC6A2 P23975 1/20 0.84
HTR2A P28223 1/20 0.84
HTR2C P28335 1/20 0.84
ADORA2A P29274 1/20 0.84
SLC6A4 P31645 1/20 0.84

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28409189 0.97 EGFR (0.86) EGFRKCNH2MLNRKDM1AABCB11
SCHEMBL17683310 0.95 EGFR (1.00) EGFRKCNH2MLNRKDM1AABCB11
SCHEMBL17553471 0.94 EGFR (1.00) EGFRKCNH2MLNRKDM1AABCB11
SCHEMBL17553693 0.94 EGFR (0.91) EGFRKCNH2MLNRKDM1AABCB11
SCHEMBL28412579 0.94 EGFR (0.91) EGFRKCNH2MLNRKDM1AABCB11
SCHEMBL22968448 0.93 EGFR (0.90) EGFRKCNH2MLNRKDM1AABCB11
SCHEMBL24117622 0.93 EGFR (0.90) EGFRKCNH2MLNRKDM1AABCB11
SCHEMBL17683220 0.93 EGFR (0.88) EGFRKCNH2MLNRKDM1AABCB11
SCHEMBL19337062 0.93 EGFR (0.87) EGFRKCNH2MLNRKDM1AABCB11
SCHEMBL17385036 0.93 EGFR (1.00) EGFRKCNH2MLNRKDM1AABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111303123-B 2- (2,4, 5-substituted anilino) pyrimidine compound and application thereof 南京雷正医药科技有限公司 2021-08-31 CN disclosed
CN-111303123-A 2- (2,4, 5-substituted anilino) pyrimidine compound and application thereof 南京雷正医药科技有限公司 2020-06-19 CN disclosed