SCHEMBL1755652

SCHEMBL1755652

CCNC(=S)Nc1ccc(-c2nc(CS(C)(=O)=O)cc(NCCO)n2)cc1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 10/20 0.48
PIK3CD O00329 10/20 0.48
MTOR P42345 5/20 0.46
CYP1A2 P05177 1/20 0.41
GPR119 Q8TDV5 1/20 0.41
JAK1 P23458 1/20 0.39
KDM4E B2RXH2 1/20 0.38
NPC1 O15118 1/20 0.38
MAPT P10636 1/20 0.38
RAB9A P51151 1/20 0.38
PIK3CB P42338 1/20 0.37
PIK3CG P48736 1/20 0.37
PTGS2 P35354 1/20 0.36
ALDH1A1 P00352 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8211495 0.83 PIK3CA (0.45) PIK3CAPIK3CDMTORCYP1A2GPR119
SCHEMBL8099679 0.83 PIK3CD (0.52) PIK3CAPIK3CDMTORJAK1KDM4E
SCHEMBL11925365 0.81 CYP1A2 (0.49) PIK3CAPIK3CDMTORCYP1A2GPR119
SCHEMBL8205211 0.79 PIK3CA (0.49) PIK3CAPIK3CDMTORCYP1A2GPR119
SCHEMBL8219095 0.79 PIK3CA (0.50) PIK3CAPIK3CDMTORCYP1A2GPR119
SCHEMBL11926810 0.77 PIK3CA (0.49) PIK3CAPIK3CDMTORCYP1A2GPR119
SCHEMBL11926789 0.77 MTOR (0.47) PIK3CAPIK3CDMTORCYP1A2GPR119
SCHEMBL11925449 0.75 CYP1A2 (0.40) PIK3CAPIK3CDMTORCYP1A2GPR119
SCHEMBL11926167 0.75 CYP1A2 (0.47) PIK3CAMTORCYP1A2GPR119PTGS2
SCHEMBL737784 0.72 PIK3CA (0.83) PIK3CAPIK3CDMTORPIK3CBPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2176238-B1 MORPHOLINO PYRIMIDINE DERIVATIVES USED IN DISEASES LINKED TO MTOR KINASE AND/OR PI3K ASTRAZENECA AB (SE) 2012-04-18 EP disclosed