SCHEMBL17558385

SCHEMBL17558385

CC(=O)Nc1cc(C(C)C2(C(C)c3ccnc(NC(C)=O)c3)NC(=O)N(c3ccc(SC(F)(F)F)cc3)C2=O)ccn1

nearest known ligand 0.56

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 19/20 0.56
LMNA P02545 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6177118 0.92 IGF1R (0.49) IGF1R
SCHEMBL6172324 0.92 IGF1R (0.47) IGF1R
SCHEMBL6174504 0.90 IGF1R (0.48) IGF1R
SCHEMBL17558370 0.89 IGF1R (0.58) IGF1R
SCHEMBL6176345 0.89 IGF1R (0.53) IGF1R
SCHEMBL6173508 0.88 IGF1R (0.56) IGF1R
SCHEMBL6173230 0.88 IGF1R (0.44) IGF1RLMNAHTT
SCHEMBL6175972 0.88 IGF1R (0.44) IGF1RLMNA
SCHEMBL6173078 0.88 IGF1R (0.45) IGF1R
SCHEMBL6175543 0.88 IGF1R (0.56) IGF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3188729-A1 CYCLIC UREA COMPOUNDS AS TROPOMYOSIN-RELATED KINASE (TRK) INHIBITORS Genzyme Corporation (US) 2017-07-12 EP disclosed
WO-2016036796-A1 CYCLIC UREA COMPOUNDS AS TROPOMYOSIN-RELATED KINASE (TRK) INHIBITORS GENZYME CORPORATION (US) 2016-03-10 WO disclosed