SCHEMBL17560422

SCHEMBL17560422

COC(=O)N1CCNC(C(N)=O)C1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.42
CHRNA4 P43681 2/20 0.42
CHRNB4 P30926 1/20 0.42
CHRNA3 P32297 1/20 0.42
TSHR P16473 1/20 0.35
SCN9A Q15858 2/20 0.34
PDE4B Q07343 4/20 0.33
PDE4A P27815 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
GAA P10253 1/20 0.33
SLC18A2 Q05940 1/20 0.31
FPR2 P25090 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.30
USP2 O75604 1/20 0.30
BIRC2 Q13490 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2C9 P11712 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14411662 0.85 CHRNB2 (0.43) CHRNB2CHRNA4CHRNB4CHRNA3TSHR
SCHEMBL28232379 0.85 MAPT (0.44) CHRNB2CHRNA4CHRNB4CHRNA3SLC18A2
SCHEMBL3561676 0.84 USP2 (0.42) PDE4BUSP2MAPT
SCHEMBL4822309 0.84 USP2 (0.42) PDE4BUSP2MAPT
SCHEMBL18129961 0.84 USP2 (0.42) PDE4BUSP2MAPT
Hydrochloric Acid SCHEMBL28060471 0.83 MAPT (0.43) CHRNB2CHRNA4CHRNB4CHRNA3SLC18A2
SCHEMBL4951081 0.82 GAA (0.37) SCN9APDE4BGAASLC18A2MAPT
SCHEMBL22220324 0.82 CHRNB2 (0.41) CHRNB2CHRNA4CHRNB4CHRNA3TSHR
SCHEMBL15432263 0.81 CHRNB2 (0.38) CHRNB2CHRNA4CHRNB4CHRNA3SCN9A
SCHEMBL7397131 0.80 SCN9A (0.34) CHRNB2CHRNA4CHRNA3SCN9AFPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016034134-A1 HETEROAROMATIC DERIVATIVES AND PHARMACEUTICAL APPLICATIONS THEREOF SUNSHINE LAKE PHARMA CO., LTD. (CN) 2016-03-10 WO disclosed